SCHEMBL3309656

SCHEMBL3309656

C=C(C)O[C@H](C(=O)O)c1c(C)cc2nc(-c3cccnc3)ccc2c1-c1ccc(Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.42
MEN1 O00255 5/20 0.42
KMT2A Q03164 5/20 0.42
MAPK1 P28482 1/20 0.42
PSD A5PKW4 2/20 0.39
POLB P06746 1/20 0.39
KDM4E B2RXH2 5/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 4/20 0.37
DHODH Q02127 2/20 0.37
HTT P42858 1/20 0.37
CYP2C9 P11712 3/20 0.37
ALDH1A1 P00352 3/20 0.37
GAA P10253 1/20 0.37
USP2 O75604 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ABL1 P00519 1/20 0.35
PDGFRB P09619 1/20 0.35
BCR P11274 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL245429 0.87 PSIP1 (0.45) MAPTMEN1KMT2AMAPK1PSD
SCHEMBL3312316 0.86 DHODH (0.33) MAPTKDM4ELMNADHODHCYP2C9
SCHEMBL3301651 0.84 CYP3A4 (0.36) KMT2APOLBKDM4EDHODHCYP3A4
SCHEMBL27928076 0.84 MEN1 (0.41) MAPTMEN1KMT2AMAPK1PSD
SCHEMBL15182573 0.83 PSD (0.40) MAPTMEN1KMT2AMAPK1PSD
SCHEMBL10284000 0.83 KMT2A (0.35) MEN1KMT2AKDM4ENPC1DHODH
SCHEMBL3295271 0.81 CYP3A4 (0.35) MAPTMEN1KMT2AMAPK1PSD
SCHEMBL10283998 0.80 EGLN1 (0.35) MAPTKMT2APOLBKDM4ELMNA
SCHEMBL3296191 0.80 GAA (0.35) MEN1KMT2AKDM4EDHODHGAA
SCHEMBL10284001 0.79 PLA2G2A (0.35) MAPTKMT2AKDM4ELMNADHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012003498-A1 2 -QUINOLINYL- ACETIC ACID DERIVATIVES AS HIV ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2012-01-05 WO disclosed