SCHEMBL3314939

SCHEMBL3314939

CCON(C(=O)[C@@H]1[C@H]2CC[C@H](C2)N1C(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C)[C@@H]1COC(=O)C1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTRA1 Q92743 1/20 0.39
CTSL P07711 2/20 0.36
ELANE P08246 2/20 0.35
CASP1 P29466 5/20 0.35
CASP3 P42574 3/20 0.35
CASP7 P55210 3/20 0.35
CASP8 Q14790 3/20 0.35
CASP6 P55212 2/20 0.35
CASP2 P42575 1/20 0.35
CASP4 P49662 1/20 0.35
CASP5 P51878 1/20 0.35
CASP9 P55211 1/20 0.35
CASP10 Q92851 1/20 0.35
CTSB P07858 2/20 0.34
CTSS P25774 2/20 0.34
CTSK P43235 2/20 0.34
CYP3A4 P08684 2/20 0.34
TSHR P16473 1/20 0.34
SYK P43405 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL993790 0.85 AGTR2 (0.37) CYP3A4
SCHEMBL3271733 0.82 CASP1 (0.43) CTSLELANECASP1CASP3CASP7
SCHEMBL1045607 0.78 CASP1 (0.36) CTSLCASP1CASP3CASP7CASP8
SCHEMBL994669 0.77 HTRA1 (0.41) HTRA1ELANECASP1CASP3CASP7
SCHEMBL13397401 0.77 HTRA1 (0.41) HTRA1ELANECASP1CASP3CASP7
SCHEMBL13528955 0.77 HTRA1 (0.41) HTRA1ELANECASP1CASP3CASP7
SCHEMBL13415945 0.77 HTRA1 (0.41) HTRA1ELANECASP1CASP3CASP7
SCHEMBL3470332 0.72 ACE (0.45) CTSLELANE
SCHEMBL7111386 0.71 ALDH1A1 (0.38) ELANECASP1CASP3CASP7CASP8
SCHEMBL5832388 0.70 CASP1 (0.45) CASP1CASP3CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100105914-A1 CASPASE INHIBITORS AND USES THEREOF VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-04-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100105914-A1 CASPASE INHIBITORS AND USES THEREOF CASP1, CASP5, CASP3 HTRA1 28/4885CTSL 37/4885ELANE 252/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.