SCHEMBL3316017

SCHEMBL3316017

C=CCOCc1cccc(C(=O)O)c1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
MRGPRX4 Q96LA9 14/20 0.53
FOLH1 Q04609 1/20 0.51
TP53 P04637 2/20 0.51
PKM P14618 2/20 0.51
NFKB1 P19838 2/20 0.51
NFKB2 Q00653 2/20 0.51
RELA Q04206 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
RAB9A P51151 2/20 0.51
RXFP1 Q9HBX9 1/20 0.51
KDM4E B2RXH2 1/20 0.51
NPC1 O15118 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isophthalic Acid SCHEMBL1360082 0.85 FFAR1 (0.51) ALDH1A1FOLH1SMN1; SMN2RAB9AKDM4E
SCHEMBL3311911 0.85 ALDH1A1 (0.52) ALDH1A1NPSR1MRGPRX4FOLH1TP53
SCHEMBL24715542 0.85 CYP3A4 (0.49) ALDH1A1NPSR1SMN1; SMN2RAB9AKDM4E
SCHEMBL6000790 0.85 MRGPRX4 (0.68) ALDH1A1NPSR1MRGPRX4FOLH1TP53
SCHEMBL28963021 0.83 FFAR1 (0.41) ALDH1A1NPSR1MRGPRX4FOLH1SMN1; SMN2
SCHEMBL27650204 0.82 NR4A2 (0.65) ALDH1A1NPSR1MRGPRX4FOLH1TP53
SCHEMBL11700680 0.81 TSHR (0.41)
SCHEMBL3314893 0.80 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2RAB9AKDM4ENPC1
SCHEMBL10653127 0.79 ALDH1A1 (0.62) ALDH1A1NPSR1MRGPRX4FOLH1TP53
SCHEMBL3315985 0.79 MRGPRX4 (0.68) ALDH1A1NPSR1MRGPRX4FOLH1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111116419-B Treprostinil intermediate and preparation process thereof 江苏豪森药业集团有限公司 2022-03-29 CN disclosed
CN-111116419-A Treprostinil intermediate and preparation process thereof 江苏豪森药业集团有限公司 2020-05-08 CN disclosed
US-8466199-B2 Allyloxy and alkyloxy benzoic acid delivery agents EMISPHERE TECHNOLOGIES, INC. (US) 2013-06-18 US disclosed
US-8466199-B2 Allyloxy and alkyloxy benzoic acid delivery agents EMISPHERE TECHNOLOGIES, INC. (US) 2013-06-18 US disclosed
US-8466199-B2 Allyloxy and alkyloxy benzoic acid delivery agents EMISPHERE TECHNOLOGIES, INC. (US) 2013-06-18 US disclosed
US-20100105604-A1 ALLYLOXY AND ALKYLOXY BENZOIC ACID DELIVERY AGENTS EMISPHERE TECHNOLOGIES, INC. (US) 2010-04-29 US disclosed
US-20100105604-A1 ALLYLOXY AND ALKYLOXY BENZOIC ACID DELIVERY AGENTS EMISPHERE TECHNOLOGIES, INC. (US) 2010-04-29 US disclosed
US-20100105604-A1 ALLYLOXY AND ALKYLOXY BENZOIC ACID DELIVERY AGENTS EMISPHERE TECHNOLOGIES, INC. (US) 2010-04-29 US disclosed
EP-2136624-A1 ALLYLQXY AND ALKYLOXY BENZOIC ACID DELIVERY AGENTS Emisphere Technologies, Inc. (US) 2009-12-30 EP disclosed
WO-2008116141-A1 ALLYLQXY AND ALKYLOXY BENZOIC ACID DELIVERY AGENTS EMISPHERE TECHNOLOGIES, INC. (US) 2008-09-25 WO disclosed
WO-2008116141-A1 ALLYLQXY AND ALKYLOXY BENZOIC ACID DELIVERY AGENTS EMISPHERE TECHNOLOGIES, INC. (US) 2008-09-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100105604-A1 ALLYLOXY AND ALKYLOXY BENZOIC ACID DELIVERY AGENTS ABCB11, TSPO, AADAC ALDH1A1 196/4885NPSR1 552/4885MRGPRX4 780/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.