Indisetron

Indisetron

SCHEMBL332330

CN1C[C@H]2C[C@@H](NC(=O)c3n[nH]c4ccccc34)C[C@@H](C1)N2C

nearest known ligand 0.83

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.61
RAB9A P51151 1/20 0.61
USP30 Q70CQ3 1/20 0.56
DYRK1A Q13627 3/20 0.55
GSK3B P49841 1/20 0.55
CHRNA7 P36544 3/20 0.55
HTR3A P46098 2/20 0.55
SMYD3 Q9H7B4 1/20 0.54
YTHDC1 Q96MU7 1/20 0.52
ALDH1A1 P00352 1/20 0.52
CYP3A4 P08684 1/20 0.52
TSHR P16473 1/20 0.52
MAPK1 P28482 1/20 0.52
HSD17B10 Q99714 1/20 0.52
RIPK1 Q13546 1/20 0.52
WNT1 P04628 1/20 0.51
HTR3E A5X5Y0 1/20 0.50
SLC22A2 O15244 1/20 0.50
HTR3B O95264 1/20 0.50
CHRNB2 P17787 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Indisetron SCHEMBL18311525 1.00 NPC1 (0.61) NPC1RAB9AUSP30DYRK1AGSK3B
Indisetron SCHEMBL1073375 1.00 NPC1 (0.61) NPC1RAB9AUSP30DYRK1AGSK3B
Indisetron SCHEMBL29398028 1.00 NPC1 (0.61) NPC1RAB9AUSP30DYRK1AGSK3B
Indisetron SCHEMBL2229963 0.99 NPC1 (0.60) NPC1RAB9AUSP30DYRK1AGSK3B
Indisetron SCHEMBL15313306 0.99 NPC1 (0.60) NPC1RAB9AUSP30DYRK1AGSK3B
Indisetron SCHEMBL2948918 0.99 NPC1 (0.60) NPC1RAB9AUSP30DYRK1AGSK3B
Indisetron SCHEMBL1649312 0.98 NPC1 (0.59) NPC1RAB9AUSP30DYRK1AGSK3B
SCHEMBL2086084 0.91 NPC1 (0.67) NPC1RAB9AUSP30DYRK1AGSK3B
SCHEMBL7336988 0.90 NPC1 (0.58) NPC1RAB9AUSP30DYRK1AGSK3B
SCHEMBL7336990 0.90 NPC1 (0.58) NPC1RAB9AUSP30DYRK1AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1644 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4602049-A1 SOS1 INHIBITORS Bayer Aktiengesellschaft (DE) 2025-08-20 EP claimed
EP-4587439-A1 SULFONE-SUBSTITUTED PYRIDO[3,4-D]PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF CANCER Bayer Aktiengesellschaft (DE) 2025-07-23 EP claimed
US-20250222003-A1 PHARMACEUTICAL COMPOSITION FOR TREATING SOLID TUMORS EISAI R&D MANAGEMENT CO., LTD. (JP) 2025-07-10 US claimed
US-20250154170-A1 FUSED PYRIMIDINES AS KRAS INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2025-05-15 US claimed
WO-2025021997-A1 NEW MAP4K1 INHIBITORS Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2025-01-30 WO claimed
WO-2025016899-A1 SPIROCYCLIC COMPOUNDS FOR THE TREATMENT OF CANCER BAYER AKTIENGESELLSCHAFT (DE) 2025-01-23 WO claimed
EP-4476221-A1 FUSED PYRIMIDINES AS KRAS INHIBITORS Bayer Aktiengesellschaft (DE) 2024-12-18 EP claimed
WO-2024188937-A1 COMBINATIONS OF ATR KINASE INHIBITORS AND PARP INHIBITORS TO TREAT HYPER-PROLIFERATIVE CONDITIONS E.G. CANCER BAYER AKTIENGESELLSCHAFT (DE) 2024-09-19 WO claimed
US-20240247015-A1 PHOSPHORUS DERIVATIVES AS NOVEL SOS1 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2024-07-25 US claimed
EP-4364742-A1 PHARMACEUTICAL COMPOSITION FOR TREATING SOLID TUMORS Eisai R&D Management Co., Ltd. (JP) 2024-05-08 EP claimed
US-6429209-B2 5-HT3 RECEPTOR ANTAGONISTS SUCH AS ALOSETRON TO TREAT NONCONSTIPATED FEMALE IRRITABLE BOWEL SYNDROME SMITHKLINE BEECHAM CORPORATION 2002-08-06 US claimed
WO-2002041918-A2 USE OF A TRIPLE COMBINATION COMPRISING A 5HT3 ANTAGONIST, A 5HT4 AGONIST AND A LAXATIVE FOR PROMOTING INTESTINAL LAVAGE JANSSEN PHARMACEUTICA N.V. (BE) 2002-05-30 WO claimed
US-20020040033-A1 Medicament containing cilansetron for the treatment of non-obstipative male irritable bowel syndrome patients SOLVAY PHARMACEUTICALS GMBH (DE) 2002-04-04 US claimed
WO-2002007713-A2 MEDICAMENTS CONTAINING CILANSETRON FOR TREATING NON-OBSTIPATED MALE IBS PATIENTS SOLVAY PHARMACEUTICALS GMBH (DE) 2002-01-31 WO claimed
US-20010044450-A1 Medicaments SEBELA INTERNATIONAL LIMITED (BM) 2001-11-22 US claimed
US-6284770-B1 ADMINISTERING SEROTONINE RECEPTOR ANTAGONIST GLAXO WELLCOME INC. 2001-09-04 US claimed
CN-1281357-A Medicaments GLAXO GROUP LTD (GB) 2001-01-24 CN claimed
EP-1021174-A2 MEDICAMENTS GLAXO GROUP LIMITED (GB) 2000-07-26 EP claimed
WO-1999017755-A2 MEDICAMENTS GLAXO GROUP LIMITED (GB) 1999-04-15 WO claimed
EP-0469449-B1 Diazabicyclononyl derivatives as 5-HT3 receptor antagonists NISSHIN FLOUR MILLING CO (JP) 1997-10-01 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250154170-A1 FUSED PYRIMIDINES AS KRAS INHIBITORS KRAS, NRAS, TP53 NPC1 3060/4885RAB9A 103/4885USP30 2092/4885
US-20010044450-A1 Medicaments HTR3A, HTR3E, HTR5A NPC1 1610/4885RAB9A 4692/4885USP30 396/4885
US-20240247015-A1 PHOSPHORUS DERIVATIVES AS NOVEL SOS1 INHIBITORS SOST, PPM1D, SOS1 NPC1 2068/4885RAB9A 1066/4885USP30 3077/4885
US-20250222003-A1 PHARMACEUTICAL COMPOSITION FOR TREATING SOLID TUMORS HTR3C, HTR3D, HTR3A NPC1 1301/4885RAB9A 779/4885USP30 3428/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.