SCHEMBL3345349

SCHEMBL3345349

COc1cc(C2CCN(CC=O)CC2)ccc1N

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
QDPR P09417 2/20 0.45
PDE4B Q07343 6/20 0.42
HTR4 Q13639 4/20 0.42
ALDH1A1 P00352 1/20 0.41
CCR5 P51681 1/20 0.41
KCNH2 Q12809 3/20 0.40
CHRM4 P08173 1/20 0.40
CHRM5 P08912 1/20 0.40
ADRA2C P18825 1/20 0.40
CHRM3 P20309 1/20 0.40
HTR1D P28221 1/20 0.40
ADRA1B P35368 1/20 0.40
HTR2B P41595 1/20 0.40
HTR3A P46098 1/20 0.40
DRD2 P14416 2/20 0.40
CARM1 Q86X55 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3345716 0.86 PDE4B (0.45) PDE4BDRD2
SCHEMBL20725583 0.84 QDPR (0.49) QDPRHTR4ALDH1A1KCNH2CHRM4
SCHEMBL15652646 0.83 QDPR (0.44) QDPRPDE4BHTR4ALDH1A1CCR5
SCHEMBL28869444 0.83 QDPR (0.48) QDPRPDE4BHTR4ALDH1A1CCR5
SCHEMBL3348766 0.82 PDE4B (0.39) QDPRPDE4BHTR4ALDH1A1
SCHEMBL310593 0.82 DRD2 (0.62) QDPRHTR4KCNH2CHRM4CHRM5
SCHEMBL2913286 0.81 HDAC1 (0.36) DRD2CARM1
SCHEMBL519815 0.81 ALK (0.51) QDPRPDE4BHTR4CCR5CHRM4
SCHEMBL520437 0.81 INSR (0.52) QDPRPDE4BCCR5DRD2
SCHEMBL310493 0.81 QDPR (0.46) QDPRHTR4KCNH2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010049731-A1 PYRAZOLO- AND IMIDAZOPYRIDINYLPYRIMIDINEAMINES AS IGF-1R TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-05-06 WO disclosed