SCHEMBL3346499

SCHEMBL3346499

CC(C)(C)Nc1cc(-c2ccc(C#Cc3ccccc3)s2)nc2ccnn12

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 7/20 0.35
CCNE1 P24864 6/20 0.35
KCNN3 Q9UGI6 6/20 0.34
KCNN1 Q92952 1/20 0.34
KCNN2 Q9H2S1 1/20 0.34
CCNT1 O60563 3/20 0.33
CDK9 P50750 3/20 0.33
CDK1 P06493 2/20 0.33
CDK4 P11802 2/20 0.33
CCNA2 P20248 2/20 0.33
CCND1 P24385 2/20 0.33
CCNA1 P78396 2/20 0.33
CDK3 Q00526 2/20 0.33
CDK7 P50613 1/20 0.33
CCNH P51946 1/20 0.33
CDK6 Q00534 1/20 0.33
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
PDE10A Q9Y233 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346921 0.90 KCNN3 (0.37) CDK2CCNE1KCNN3CCNT1CDK9
SCHEMBL3348362 0.90 CDK2 (0.39) CDK2CCNE1
SCHEMBL3351713 0.89 KCNN3 (0.38) CDK2CCNE1KCNN3KCNN1KCNN2
SCHEMBL3345910 0.89 GRM5 (0.35) CDK2CCNE1CCNT1CDK9CDK1
SCHEMBL3351751 0.87 CDK2 (0.38) CDK2CCNE1KCNN3KCNN1KCNN2
SCHEMBL3351298 0.87 GRM5 (0.33)
SCHEMBL3347648 0.87 GRM5 (0.33) CDK2CCNE1KCNN3KCNN1KCNN2
SCHEMBL3346746 0.87 KCNN1 (0.38) CDK2CCNE1KCNN3KCNN1KCNN2
SCHEMBL3347209 0.86 KCNN3 (0.36) CDK2CCNE1KCNN3KCNN1KCNN2
SCHEMBL3347564 0.86 GRM5 (0.33) CDK2CCNE1KCNN3CCNT1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO claimed
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed