SCHEMBL3346746

SCHEMBL3346746

CC(C)(C)Nc1cc(-c2ccc(C#Cc3cccs3)s2)nc2ccnn12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN1 Q92952 1/20 0.38
KCNN2 Q9H2S1 1/20 0.38
KCNN3 Q9UGI6 1/20 0.38
PIM1 P11309 2/20 0.34
PIM3 Q86V86 1/20 0.34
PLK3 Q9H4B4 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
GRM5 P41594 2/20 0.33
GSK3B P49841 2/20 0.33
AURKA O14965 1/20 0.33
JAK2 O60674 1/20 0.33
NTRK1 P04629 1/20 0.33
RET P07949 1/20 0.33
FGFR1 P11362 1/20 0.33
PRKACA P17612 1/20 0.33
LTK P29376 1/20 0.33
KDR P35968 1/20 0.33
MAP2K2 P36507 1/20 0.33
FLT3 P36888 1/20 0.33
MAPK8 P45983 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346499 0.87 CDK2 (0.35) KCNN1KCNN2KCNN3CDK5CDK2
SCHEMBL3347071 0.85 CYP2A6 (0.32) KCNN1KCNN2KCNN3CDK5CDK2
SCHEMBL3347648 0.84 GRM5 (0.33) KCNN1KCNN2KCNN3GRM5CDK2
SCHEMBL3351751 0.84 CDK2 (0.38) KCNN1KCNN2KCNN3GRM5CDK5
SCHEMBL3351298 0.84 GRM5 (0.33) GRM5
SCHEMBL3348362 0.83 CDK2 (0.39) GRM5CDK2CCNE1
SCHEMBL3345946 0.83 GRM5 (0.39) KCNN3GRM5CDK2KDM4EALDH1A1
SCHEMBL3346921 0.83 KCNN3 (0.37) KCNN3GRM5CDK2CCNE1CCNT1
SCHEMBL3346510 0.83 GRM5 (0.37) GRM5PDE10A
SCHEMBL3347209 0.83 KCNN3 (0.36) KCNN1KCNN2KCNN3GRM5CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO claimed
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed