SCHEMBL3346856

SCHEMBL3346856

Cc1cccc(C#CCCc2ccn3nc(C)cc3n2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 19/20 0.52
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
PKM P14618 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
CYP2C19 P33261 1/20 0.37
THPO P40225 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
GRIN2B Q13224 1/20 0.37
GRM1 Q13255 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346938 0.89 GRM5 (0.43) GRM5KDM4EALDH1A1MAPK1HTT
SCHEMBL3347055 0.86 GRM5 (0.51) GRM5KDM4EALDH1A1CYP1A2MAPK1
SCHEMBL3345876 0.84 GRM5 (0.53) GRM5KDM4EALDH1A1MEN1NPC1
SCHEMBL3351704 0.83 KDM4E (0.34) GRM5KDM4EALDH1A1MAPK1HTT
SCHEMBL3345928 0.83 GRM5 (0.36) GRM5KDM4EALDH1A1MEN1NPC1
SCHEMBL3347641 0.82 GRM5 (0.38) GRM5KDM4EALDH1A1SMN1; SMN2MAPK1
SCHEMBL3345927 0.81 GRM5 (0.36) GRM5CYP1A2CYP2D6
SCHEMBL3347285 0.81 KDM4E (0.37) KDM4EALDH1A1MAPK1HTTL3MBTL1
SCHEMBL3351706 0.81 KDM4E (0.34) GRM5KDM4EALDH1A1MAPK1HTT
SCHEMBL3345594 0.81 GRM5 (0.40) GRM5KDM4EALDH1A1MAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed