SCHEMBL3348606

SCHEMBL3348606

O=C1C=CC2=Nc3ccccc3C2=C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.38
MAOB P27338 3/20 0.38
HSD17B3 P37058 1/20 0.36
MEN1 O00255 4/20 0.34
KMT2A Q03164 4/20 0.34
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 3/20 0.34
LMNA P02545 3/20 0.34
MAPT P10636 3/20 0.34
HKDC1 Q2TB90 2/20 0.34
APAF1 O14727 2/20 0.34
GALK1 P51570 2/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
TSHR P16473 1/20 0.34
HK1 P19367 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CDC25B P30305 3/20 0.33
IDO1 P14902 3/20 0.33
AKT1 P31749 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30804593 1.00 MAOA (0.38) MAOAMAOBHSD17B3MEN1KMT2A
SCHEMBL30483749 0.78 MAOA (0.36) MAOAMAOBCDC25B
SCHEMBL29593696 0.75 MEN1 (0.31) MEN1KMT2A
SCHEMBL4739721 0.74 KDM4E (0.33) MEN1KMT2AALDH1A1KDM4ELMNA
SCHEMBL1758940 0.72 IDO1 (0.33) IDO1
SCHEMBL30997931 0.69 MAPT (0.38) MAOAMAOBMEN1KMT2AALDH1A1
SCHEMBL536721 0.69 MAPT (0.38) MAOAMAOBMEN1KMT2AALDH1A1
SCHEMBL27798673 0.69 IDO1 (0.32) IDO1
SCHEMBL1357123 0.68 IDO1 (0.31) IDO1
SCHEMBL7675144 0.68 IDO1 (0.31) IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007047579-A2 A NOVEL THERAPEUTIC TARGET FOR PROTOZOAL DISEASES VIRGINIA TECH INTELLECTUAL PROPERTIES, INC. (US) 2007-04-26 WO claimed
US-5801190-A Fused pyrrolo 2,3-C! carbazole-6-ones CEPHALON, INC. (US) 1998-09-01 US claimed
CN-117616032-A Rare earth complex 东曹株式会社 2024-02-27 CN disclosed
US-11377415-B2 Method for converting N,N-dialkylamide compound into ester compound using complex of fourth-period transition metal as catalyst TAKASAGO INTERNATIONAL CORPORATION (JP) 2022-07-05 US disclosed
EP-3760607-A1 METHOD FOR CONVERTING N,N-DIALKYLAMIDE COMPOUND INTO ESTER COMPOUND USING COMPLEX OF FOURTH-PERIOD TRANSITION METAL AS CATALYST Takasago International Corporation (JP) 2021-01-06 EP disclosed
US-20200399200-A1 METHOD FOR CONVERTING N,N-DIALKYLAMIDE COMPOUND INTO ESTER COMPOUND USING COMPLEX OF FOURTH-PERIOD TRANSITION METAL AS CATALYST TAKASAGO INTERNATIONAL CORPORATION (JP) 2020-12-24 US disclosed
WO-2010042445-A1 CARBAZOLE COMPOUNDS AND THERAPEUTIC USES OF THE COMPOUNDS CLEVELAND BIOLABS, INC. (US) 2010-04-15 WO disclosed
US-6821644-B2 BIS(DIARYLAMINO)ARYLENE COMPOUND; BRILLIANCE, DURABILITY SAMSUNG SDI CO., LTD. (KR) 2004-11-23 US disclosed
CN-1098266-C Fused pyrrolo (2,3-C) carbazole-6-ones which potentiate activity of gamma interferon CEPHALON INC (US) 2003-01-08 CN disclosed
CN-1098266-C Fused pyrrolo (2,3-C) carbazole-6-ones which potentiate activity of gamma interferon CEPHALON INC (US) 2003-01-08 CN disclosed
EP-0885229-B1 FUSED PYRROLO(2,3-C)CARBAZOLE-6-ONES WHICH POTENTIATE ACTIVITY OF GAMMA INTERFERON CEPHALON INC (US) 2000-08-02 EP disclosed
CN-1211254-A Fused pyrrolo (2,3-C) carbazole-6-ones which potentiate activity of gamma interferon CEPHALON INC (US) 1999-03-17 CN disclosed
CN-1211254-A Fused pyrrolo (2,3-C) carbazole-6-ones which potentiate activity of gamma interferon CEPHALON INC (US) 1999-03-17 CN disclosed
EP-0885229-A1 FUSED PYRROLO(2,3-C)CARBAZOLE-6-ONES WHICH POTENTIATE ACTIVITY OF GAMMA INTERFERON CEPHALON, INC. (US) 1998-12-23 EP disclosed
US-5801190-A Fused pyrrolo 2,3-C! carbazole-6-ones CEPHALON, INC. (US) 1998-09-01 US disclosed
US-5801190-A Fused pyrrolo 2,3-C! carbazole-6-ones CEPHALON, INC. (US) 1998-09-01 US disclosed
US-5801190-A Fused pyrrolo 2,3-C! carbazole-6-ones CEPHALON, INC. (US) 1998-09-01 US disclosed
WO-1997031002-A9 FUSED PYRROLO(2,3-C)CARBAZOLE-6-ONES WHICH POTENTIATE ACTIVITY OF GAMMA INTERFERON 1997-10-30 WO disclosed
WO-1997031002-A1 FUSED PYRROLO(2,3-C)CARBAZOLE-6-ONES WHICH POTENTIATE ACTIVITY OF GAMMA INTERFERON CEPHALON, INC. (US) 1997-08-28 WO disclosed
US-5616724-A FOR POTENTIATION OF HUMAN INTERFERON-GAMMA; IMMUNOLOGY CEPHALON, INC. (US) 1997-04-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11377415-B2 Method for converting N,N-dialkylamide compound into ester compound using complex of fourth-period transition metal as catalyst NEK4, TENT4A, TCF4 MAOA 2320/4885MAOB 2240/4885HSD17B3 2623/4885
US-20200399200-A1 METHOD FOR CONVERTING N,N-DIALKYLAMIDE COMPOUND INTO ESTER COMPOUND USING COMPLEX OF FOURTH-PERIOD TRANSITION METAL AS CATALYST NEK4, TENT4A, TCF4 MAOA 2320/4885MAOB 2240/4885HSD17B3 2623/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.