SCHEMBL3351536

SCHEMBL3351536

CC(=O)C(Cc1ccc(S(C)(=O)=O)cc1)C(O)=S

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.41
ITGA4 P13612 1/20 0.41
LDHA P00338 1/20 0.39
ENPP2 Q13822 1/20 0.39
AKR1C3 P42330 1/20 0.39
GSR P00390 2/20 0.39
KDM4E B2RXH2 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
LMNA P02545 1/20 0.37
PTGS2 P35354 3/20 0.37
EPHX2 P34913 1/20 0.37
NR1H4 Q96RI1 1/20 0.37
EPHX1 P07099 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
GRM4 Q14833 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3787450 0.89 ENPP2 (0.45) ITGB1ITGA4LDHAENPP2AKR1C3
SCHEMBL15647871 0.83 LDHA (0.55) ITGB1ITGA4LDHAENPP2AKR1C3
SCHEMBL3351530 0.83 ENPP2 (0.40) ITGB1ITGA4LDHAENPP2AKR1C3
SCHEMBL534070 0.81 ENPP2 (0.39) ITGB1ITGA4ENPP2AKR1C3SMN1; SMN2
SCHEMBL7274800 0.80 MDM2 (0.53) LMNA
SCHEMBL7274790 0.80 MDM2 (0.53) LMNA
SCHEMBL3772833 0.79 MMP8 (0.47)
SCHEMBL27801725 0.79 MME (0.43) LDHAEPHX1
SCHEMBL4634330 0.77 LMNA (0.44) ITGB1ITGA4AKR1C3LMNAEPHX2
SCHEMBL3785349 0.77 EPHX2 (0.39) ITGB1ITGA4ENPP2AKR1C3GSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010040989-A1 QUINOLIN-2-ONE COMPOUNDS ARGENTA ORAL THERAPEUTICS LIMITED (GB) 2010-04-15 WO disclosed