SCHEMBL335570

SCHEMBL335570

Nc1nc2ccc(NC(=O)C(O)C(NC(=O)c3cc4ccccc4s3)c3ccccc3)cc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 6/20 0.47
HDAC1 Q13547 5/20 0.42
ACP1 P24666 1/20 0.40
APP P05067 1/20 0.40
TMIGD3 P0DMS9 1/20 0.39
ADORA1 P30542 1/20 0.39
STAT1 P42224 1/20 0.39
CASP3 P42574 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
MCHR1 Q99705 1/20 0.39
ABL1 P00519 1/20 0.39
FABP6 P51161 1/20 0.39
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL335244 0.89 MAPT (0.41) PIN1HDAC1ACP1ABL1FABP6
SCHEMBL335890 0.85 ACP1 (0.40) PIN1HDAC1ACP1ABL1FABP6
SCHEMBL15282285 0.85 ACP1 (0.46) ACP1ABL1FABP6MAPTRAB9A
SCHEMBL15282212 0.85 ACP1 (0.46) ACP1ABL1FABP6MAPTRAB9A
SCHEMBL334912 0.84 F7 (0.40) PIN1HDAC1ACP1ABL1FABP6
SCHEMBL335286 0.84 ACP1 (0.42) ACP1CASP3SENP8SENP7SENP6
SCHEMBL335351 0.84 EGFR (0.50) HDAC1ACP1APPABL1FABP6
SCHEMBL335390 0.84 ABL1 (0.44) PIN1ACP1ABL1FABP6MAPT
SCHEMBL335694 0.84 SMN1; SMN2 (0.39) PIN1HDAC1ACP1ABL1FABP6
SCHEMBL336367 0.84 MAPT (0.47) ACP1ABL1FABP6MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8097758-B2 Isoserine derivatives for use as coagulation factor IXa inhibitors SANOFI-AVENTIS (FR) 2012-01-17 US claimed