SCHEMBL3362275

SCHEMBL3362275

NS(=O)(=O)c1ccccc1CN1CCOCC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A13 Q16696 5/20 0.59
KMT2A Q03164 3/20 0.47
CYP2C9 P11712 2/20 0.47
ALDH1A1 P00352 2/20 0.47
MEN1 O00255 2/20 0.47
ALOX15 P16050 1/20 0.47
HSD17B10 Q99714 1/20 0.47
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
CTSB P07858 1/20 0.45
CA2 P00918 4/20 0.44
ADORA2A P29274 1/20 0.44
ADORA1 P30542 1/20 0.44
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
CA1 P00915 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21962272 0.88 CYP2A13 (0.53) CYP2A13KMT2ACYP2C9ALDH1A1MEN1
SCHEMBL10642464 0.85 ALDH1A1 (0.50) KMT2ACYP2C9ALDH1A1MEN1CYP3A4
SCHEMBL5251939 0.85 KMT2A (0.49) CYP2A13KMT2AALDH1A1MEN1CA2
SCHEMBL28532123 0.84 CYP2A13 (0.55) CYP2A13KMT2ACYP2C9ALDH1A1MEN1
SCHEMBL4441883 0.81 CYP2A13 (0.55) CYP2A13KMT2AALDH1A1MEN1CA2
SCHEMBL11193326 0.79 CYP2A13 (0.75) CYP2A13KMT2ACYP2C9ALDH1A1MEN1
SCHEMBL22501227 0.77 MAPT (0.51) KMT2AALDH1A1MEN1CA2KDM4E
SCHEMBL31680437 0.75 CA2 (0.42) CYP2A13CYP2C9ALDH1A1CYP3A4CYP2D6
SCHEMBL4100083 0.75 CYP2A13 (1.00) CYP2A13KMT2ACYP2C9ALDH1A1MEN1
SCHEMBL4327006 0.75 MPO (0.75) CYP2A13KMT2ACYP2C9ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100009970-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF VIRAL DISEASES COMBINATORX (SINGAPORE) PTE. LTD. (SG) 2010-01-14 US disclosed
EP-2094670-A1 HETEROCYCLYC SULFONAMIDES HAVING EDG-I ANTAGONISTIC ACTIVITY AstraZeneca AB (SE) 2009-09-02 EP disclosed
WO-2008056150-A1 HETEROCYCLYC SULFONAMIDES HAVING EDG-I ANTAGONISTIC ACTIVITY ASTRAZENECA AB (SE) 2008-05-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100009970-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF VIRAL DISEASES HTR1A, HTR3B, HTR3A CYP2A13 593/4885KMT2A 1108/4885CYP2C9 1449/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.