SCHEMBL3364589

SCHEMBL3364589

Cn1nc2c(-c3ccccc3Oc3ccccc3)cccc2c1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 14/20 0.44
SCN9A Q15858 1/20 0.40
SCN1A P35498 1/20 0.38
SCN2A Q99250 1/20 0.38
SCN3A Q9NY46 1/20 0.38
PTGS2 P35354 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3364448 0.89 BRD4 (0.47) BRD4SCN9ASCN1ASCN2ASCN3A
SCHEMBL3368049 0.85 DHODH (0.41) SCN9A
SCHEMBL3365087 0.80 BRD4 (0.43) BRD4SCN9A
SCHEMBL3365869 0.80 CYP3A4 (0.40) BRD4
SCHEMBL3362827 0.77 GABRG2 (0.50)
SCHEMBL3365574 0.77 BRD4 (0.47) BRD4
SCHEMBL3364893 0.75 SMN1; SMN2 (0.40) SCN9A
SCHEMBL3364109 0.73 GABRG2 (0.41)
SCHEMBL3367536 0.72 CRHR1 (0.49)
SCHEMBL3366144 0.72 ALDH1A1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656353-B1 GABANERGIC MODULATORS HOFFMANN LA ROCHE (CH) 2010-01-27 EP claimed