SCHEMBL3365574

SCHEMBL3365574

COc1cccc(-c2cccc3c(C(=O)O)n(C)nc23)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.47
LMNA P02545 2/20 0.45
MAPK1 P28482 1/20 0.45
ALDH1A1 P00352 2/20 0.44
HPGD P15428 1/20 0.44
RECQL P46063 1/20 0.44
PRKAB2 O43741 1/20 0.43
PRKAG1 P54619 1/20 0.43
PRKAA2 P54646 1/20 0.43
PRKAA1 Q13131 1/20 0.43
PRKAG3 Q9UGI9 1/20 0.43
PRKAG2 Q9UGJ0 1/20 0.43
PRKAB1 Q9Y478 1/20 0.43
NR1H2 P55055 1/20 0.43
NR1H3 Q13133 1/20 0.43
KMT2A Q03164 1/20 0.42
GRIA2 P42262 1/20 0.42
GRIA4 P48058 1/20 0.42
PIN1 Q13526 1/20 0.42
GPR35 Q9HC97 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3364994 0.89 BRD4 (0.46) BRD4LMNAMAPK1ALDH1A1HPGD
SCHEMBL3365869 0.84 CYP3A4 (0.40) BRD4ALDH1A1HPGDKMT2AKDM4E
SCHEMBL3365166 0.84 GABRG2 (0.42) KMT2AGRIA2GRIA4PIN1MCL1
SCHEMBL3362827 0.83 GABRG2 (0.50) ALDH1A1HPGDKMT2AMAPT
SCHEMBL3367525 0.83 KMT2A (0.48) ALDH1A1KMT2AKDM4ESMN1; SMN2
SCHEMBL3368049 0.81 DHODH (0.41) MCL1
SCHEMBL3365908 0.80 BRD4 (0.44) BRD4LMNAMAPK1ALDH1A1HPGD
SCHEMBL3364109 0.80 GABRG2 (0.41) ALDH1A1HPGDKDM4EMAPT
SCHEMBL3364589 0.77 BRD4 (0.44) BRD4
SCHEMBL27359949 0.77 BRD4 (0.45) BRD4ALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656353-B1 GABANERGIC MODULATORS HOFFMANN LA ROCHE (CH) 2010-01-27 EP claimed