SCHEMBL3368049

SCHEMBL3368049

Cn1nc2c(-c3ccc(Oc4ccccc4)cc3)cccc2c1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.41
GSTP1 P09211 1/20 0.40
SCN4A P35499 1/20 0.40
MGLL Q99685 1/20 0.39
PPARG P37231 5/20 0.39
PPARA Q07869 5/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
PPARD Q03181 1/20 0.39
SCN9A Q15858 3/20 0.38
MCL1 Q07820 3/20 0.38
CYSLTR1 Q9Y271 1/20 0.38
BCL2 P10415 2/20 0.38
MDM2 Q00987 2/20 0.38
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3364893 0.89 SMN1; SMN2 (0.40) GSTP1SCN4AMGLLPPARGPPARA
SCHEMBL3365869 0.88 CYP3A4 (0.40) DHODHCYP2C9
SCHEMBL3364589 0.85 BRD4 (0.44) SCN9A
SCHEMBL3365574 0.81 BRD4 (0.47) MCL1
SCHEMBL3367042 0.81 DHODH (0.41) DHODHPPARGPPARACYP2C9
SCHEMBL3364363 0.80 HSP90AA1 (0.41) GSTP1SCN4AMGLLPPARGPPARA
SCHEMBL14231105 0.80 GSTP1 (0.40) GSTP1SCN4AMGLLPPARGPPARA
SCHEMBL3364109 0.78 GABRG2 (0.41)
SCHEMBL3365166 0.77 GABRG2 (0.42) DHODHMCL1
SCHEMBL3363948 0.76 GPR35 (0.40) DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656353-B1 GABANERGIC MODULATORS HOFFMANN LA ROCHE (CH) 2010-01-27 EP claimed