SCHEMBL3365166

SCHEMBL3365166

Cc1cccc(-c2cccc3c(C(=O)O)n(C)nc23)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42
GABRA2 P47869 1/20 0.42
ENPP1 P22413 1/20 0.41
KMO O15229 2/20 0.40
RPA1 P27694 2/20 0.40
CNR2 P34972 1/20 0.39
PIN1 Q13526 1/20 0.39
LDHA P00338 1/20 0.39
LDHB P07195 1/20 0.39
MCL1 Q07820 3/20 0.39
BAD Q92934 3/20 0.39
KMT2A Q03164 1/20 0.39
GRIA2 P42262 1/20 0.38
GRIA4 P48058 1/20 0.38
F11 P03951 1/20 0.38
IP6K1 Q92551 1/20 0.38
IP6K3 Q96PC2 1/20 0.38
IP6K2 Q9UHH9 1/20 0.38
FBP1 P09467 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3364109 0.91 GABRG2 (0.41) GABRG2GABRB3GABRA2KMORPA1
SCHEMBL3365869 0.88 CYP3A4 (0.40) GABRG2GABRB3GABRA2ENPP1CNR2
SCHEMBL3364407 0.86 HSD17B10 (0.44) GABRG2GABRB3GABRA2ENPP1KMT2A
SCHEMBL3365574 0.84 BRD4 (0.47) PIN1MCL1BADKMT2AGRIA2
SCHEMBL4700361 0.82 CRHR1 (0.40) GABRG2GABRB3GABRA2MCL1KMT2A
SCHEMBL18512112 0.78 CYP1A2 (0.43) KMT2A
SCHEMBL3363948 0.78 GPR35 (0.40) GABRG2GABRB3GABRA2ENPP1DHODH
SCHEMBL3368008 0.78 HRH4 (0.43)
SCHEMBL3367042 0.78 DHODH (0.41) KMT2ADHODH
SCHEMBL14231320 0.77 ENPP1 (0.42) GABRG2GABRB3GABRA2ENPP1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656353-B1 GABANERGIC MODULATORS HOFFMANN LA ROCHE (CH) 2010-01-27 EP claimed