SCHEMBL3365908

SCHEMBL3365908

COC(=O)Oc1c2cccc(-c3cccc(OC)c3)c2nn1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.44
HSP90AA1 P07900 1/20 0.43
HSP90AB1 P08238 1/20 0.43
TP53 P04637 3/20 0.41
DGAT2 Q96PD7 4/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.40
PIK3CG P48736 1/20 0.40
MAPT P10636 3/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 1/20 0.39
LMNA P02545 2/20 0.39
GPR84 Q9NQS5 1/20 0.39
ALDH1A1 P00352 2/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ADORA3 P0DMS8 1/20 0.39
ADORA2B P29275 1/20 0.39
ADORA1 P30542 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3364346 0.87 GABRG2 (0.43) HSD17B10KMT2A
SCHEMBL3365864 0.84 CRHR1 (0.44) KDM4ELMNAALDH1A1SMN1; SMN2ADORA3
SCHEMBL3368213 0.84 GABRG2 (0.51) LMNAALDH1A1SMN1; SMN2ADORA3MEN1
SCHEMBL3363718 0.84 GABRG2 (0.42) MAPTHPGDLMNAALDH1A1SMN1; SMN2
SCHEMBL3364363 0.83 HSP90AA1 (0.41) HSP90AA1HSP90AB1MAPK1SMN1; SMN2
SCHEMBL3364994 0.81 BRD4 (0.46) BRD4HSP90AA1HSP90AB1TP53DGAT2
SCHEMBL3365035 0.81 TP53 (0.39) TP53MAPTKDM4EHPGDALDH1A1
SCHEMBL3365574 0.80 BRD4 (0.47) BRD4DGAT2TSHRMAPK1MAPT
SCHEMBL3368191 0.80 TUBB4A (0.38) PIK3CGMAPTKDM4EHSD17B10MEN1
SCHEMBL3362490 0.80 HRH4 (0.40) MAPK1GPR84ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656353-B1 GABANERGIC MODULATORS HOFFMANN LA ROCHE (CH) 2010-01-27 EP claimed