SCHEMBL3365883

SCHEMBL3365883

N#Cc1ccc(-c2ccnc(Cl)c2)c(C(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.50
AKR1C2 P52895 1/20 0.50
TRPV4 Q9HBA0 1/20 0.47
AR P10275 6/20 0.43
KIF11 P52732 1/20 0.39
S1PR1 P21453 1/20 0.38
S1PR3 Q99500 1/20 0.38
NSD2 O96028 1/20 0.38
PARP10 Q53GL7 1/20 0.37
PARP11 Q9NR21 1/20 0.37
EGLN2 Q96KS0 1/20 0.37
AAK1 Q2M2I8 1/20 0.37
PTGS2 P35354 2/20 0.36
GRM5 P41594 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3362974 0.83 S1PR1 (0.47) TRPV4ARKIF11S1PR1S1PR3
SCHEMBL3362125 0.81 EGLN2 (0.50) ARPARP10PARP11EGLN2GRM5
SCHEMBL28668535 0.77 KIF11 (0.57) TRPV4ARKIF11NSD2
SCHEMBL7604551 0.77 TRPV4 (0.56) TRPV4ARKIF11NSD2
SCHEMBL23994244 0.76 AKR1C3 (0.50) AKR1C3AKR1C2ARS1PR1S1PR3
SCHEMBL30224509 0.76 AKR1C3 (0.50) AKR1C3AKR1C2ARS1PR1S1PR3
SCHEMBL1934802 0.75 GRM2 (0.43) AKR1C3AKR1C2ARGRM5
SCHEMBL2371259 0.74 AR (0.47) TRPV4ARKIF11S1PR1S1PR3
SCHEMBL2743433 0.74 MAPKAPK2 (0.48) KIF11EGLN2GRM5
SCHEMBL249837 0.73 CYP11B2 (0.54) TRPV4ARS1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed