SCHEMBL3362974

SCHEMBL3362974

N#Cc1ccc(-c2ccnc(N)c2)c(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.47
S1PR3 Q99500 1/20 0.47
PDE3B Q13370 1/20 0.47
PDE3A Q14432 1/20 0.47
AR P10275 5/20 0.43
DYRK1A Q13627 2/20 0.42
GSK3B P49841 1/20 0.41
NOS3 P29474 1/20 0.41
NOS2 P35228 1/20 0.41
TRPV4 Q9HBA0 1/20 0.40
CDC7 O00311 1/20 0.40
CDK2 P24941 1/20 0.40
NSD2 O96028 1/20 0.40
KIF11 P52732 1/20 0.39
AAK1 Q2M2I8 1/20 0.39
ALOX5AP P20292 2/20 0.38
FEN1 P39748 2/20 0.38
AKT1 P31749 1/20 0.38
PIK3CA P42336 1/20 0.38
MTOR P42345 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3365883 0.83 AKR1C3 (0.50) S1PR1S1PR3ARTRPV4NSD2
SCHEMBL3360845 0.78 EGLN2 (0.48) ARDYRK1AGSK3BCDC7CDK2
SCHEMBL3366217 0.78 KCNH2 (0.52) S1PR1DYRK1AGSK3BNOS3NOS2
SCHEMBL28668535 0.77 KIF11 (0.57) ARTRPV4NSD2KIF11
SCHEMBL7604551 0.77 TRPV4 (0.56) ARTRPV4NSD2KIF11GLA
SCHEMBL3393608 0.76 BACE1 (0.56) S1PR1S1PR3PDE3BPDE3AAR
SCHEMBL2371259 0.74 AR (0.47) S1PR1S1PR3ARTRPV4KIF11
SCHEMBL3397985 0.74 DYRK1A (0.54) DYRK1AGSK3BCDC7CDK2AAK1
SCHEMBL29432635 0.74 DYRK1A (0.54) DYRK1AGSK3BCDC7CDK2AAK1
SCHEMBL249837 0.73 CYP11B2 (0.54) S1PR1PDE3BPDE3AARTRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed