SCHEMBL3363718

SCHEMBL3363718

COC(=O)Oc1c2cccc(-c3cc(C)cc(C)c3)c2nn1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 2/20 0.42
GABRB3 P28472 2/20 0.42
GABRA2 P47869 2/20 0.42
CHRM3 P20309 3/20 0.37
BRD9 Q9H8M2 1/20 0.36
BRD7 Q9NPI1 1/20 0.36
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
F2 P00734 1/20 0.32
PLAU P00749 1/20 0.32
ELANE P08246 1/20 0.32
HPGD P15428 2/20 0.32
KDR P35968 2/20 0.32
KCNT1 Q5JUK3 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3364346 0.92 GABRG2 (0.43) GABRG2GABRB3GABRA2CHRM3F2
SCHEMBL28759985 0.88 GABRG2 (0.41) GABRG2GABRB3GABRA2CHRM3BRD9
SCHEMBL3365908 0.84 BRD4 (0.44) MAPTHPGDSMN1; SMN2ALDH1A1LMNA
SCHEMBL3365035 0.82 TP53 (0.39) MAPTHPGDSMN1; SMN2ALDH1A1
SCHEMBL3362490 0.81 HRH4 (0.40) ELANEALDH1A1
SCHEMBL3368191 0.81 TUBB4A (0.38) MAPTPLAUELANEKDR
SCHEMBL3364428 0.81 GABRG2 (0.41) GABRG2GABRB3GABRA2CHRM3BRD9
SCHEMBL3364363 0.81 HSP90AA1 (0.41) SMN1; SMN2
SCHEMBL3364228 0.78 CRHR1 (0.46) CNR1CNR2HPGDALDH1A1
SCHEMBL3367673 0.78 S1PR4 (0.38) HPGDSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656353-B1 GABANERGIC MODULATORS HOFFMANN LA ROCHE (CH) 2010-01-27 EP claimed