SCHEMBL3373429

SCHEMBL3373429

Nc1ccc(C(=O)CO)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.47
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 2/20 0.47
MAOA P21397 1/20 0.47
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
CYP19A1 P11511 2/20 0.46
MAPT P10636 4/20 0.45
KDM4E B2RXH2 2/20 0.45
HIF1A Q16665 1/20 0.45
SLC22A6 Q4U2R8 1/20 0.45
SLC22A8 Q8TCC7 1/20 0.45
APEX1 P27695 3/20 0.45
POLB P06746 2/20 0.45
TDP1 Q9NUW8 2/20 0.45
PKM P14618 1/20 0.45
PARP10 Q53GL7 1/20 0.43
MASP2 O00187 1/20 0.42
PLAU P00749 1/20 0.42
THPO P40225 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29131268 0.91 RAB9A (0.45) LMNACYP1A2CYP3A4MAOAMEN1
SCHEMBL29122221 0.91 LMNA (0.41) LMNACYP1A2CYP3A4MAOAMEN1
SCHEMBL30694356 0.87 KDM4E (0.50) CYP3A4MEN1KMT2AMAPTKDM4E
SCHEMBL11365527 0.82 MAPT (0.56) LMNACYP1A2CYP3A4MAOAMEN1
SCHEMBL7343185 0.81 TDP1 (0.65) LMNACYP1A2CYP3A4MAOAMEN1
SCHEMBL9547546 0.80 LMNA (0.47) LMNACYP1A2CYP3A4MAOAMEN1
SCHEMBL3181886 0.80 LMNA (0.47) LMNACYP1A2CYP3A4MAOAMEN1
SCHEMBL3376212 0.80 PARP10 (0.50) CYP3A4KMT2AMAPTPOLBTDP1
SCHEMBL221282 0.78 MAPT (0.57) LMNACYP1A2CYP3A4MAOAMEN1
SCHEMBL2151966 0.78 GSK3B (0.64) LMNACYP1A2CYP3A4MAOAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 55 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109169659-B Application of 4-amino-2-hydroxyacetophenone in preparation of pesticide for resisting agrobacterium infection 南京理工大学 2020-12-04 CN claimed
CN-104311567-B One prepares the method for 4-amino-3-(4-amino-benzene) furo [2,3-d] pyrimidine SHANGHAI INSTITUTE OF TECHNOLOGY (CN) 2016-04-27 CN claimed
EP-2507243-B1 SPIROINDOLINONE PYRROLIDINES HOFFMANN LA ROCHE (CH) 2015-06-10 EP claimed
CN-104311567-A Method for preparing 4-amino-3-(4-aminobenzene)furo[2,3-d] pyrimidine SHANGHAI INST TECHNOLOGY 2015-01-28 CN claimed
US-8354444-B2 Substituted pyrrolidine-2-carboxamides HOFFMANN-LA ROCHE INC. (US) 2013-01-15 US claimed
EP-2507243-A1 SPIROINDOLINONE PYRROLIDINES F. Hoffmann-La Roche AG (CH) 2012-10-10 EP claimed
US-20100152190-A1 Substituted Pyrrolidine-2-Carboxamides F. HOFFMANN-LA ROCHE AG (CH) 2010-06-17 US claimed
US-20100075948-A1 Substituted Pyrrolidine-2-Carboxamides DING QINGJIE 2010-03-25 US claimed
EP-0011490-B2 ANALGESIC TABLET AND PROCESS FOR ITS PREPARATION BEECHAM GROUP PLC (GB) 1989-10-18 EP claimed
EP-0011490-B1 ANALGESIC TABLET AND PROCESS FOR ITS PREPARATION BEECHAM GROUP PLC (GB) 1982-11-03 EP claimed
US-11332389-B1 Recylable multifunctional composites for metal ion removal from water KING ABDULAZIZ UNIVERSITY (SA) 2022-05-17 US disclosed
CN-109169659-B Application of 4-amino-2-hydroxyacetophenone in preparation of pesticide for resisting agrobacterium infection 南京理工大学 2020-12-04 CN disclosed
CN-109169659-B Application of 4-amino-2-hydroxyacetophenone in preparation of pesticide for resisting agrobacterium infection 南京理工大学 2020-12-04 CN disclosed
CN-109169659-B Application of 4-amino-2-hydroxyacetophenone in preparation of pesticide for resisting agrobacterium infection 南京理工大学 2020-12-04 CN disclosed
EP-2534132-B1 SUBSTITUTED PYRROLIDINE-2-CARBOXAMIDES HOFFMANN LA ROCHE (CH) 2017-04-26 EP disclosed
US-4479007-A Chroman-4-ones and process for preparing same BAYER AKTIENGESELLSCHAFT (DE) 1984-10-23 US disclosed
US-4415741-A REACTING O-HYDROXYACETOPHENONE AND CYCLOPENTANONE BAYER AKTIENGESELLSCHAFT (DE) 1983-11-15 US disclosed
EP-0013879-B1 REACTIVE DYESTUFFS, THEIR PREPARATION AND THEIR USE FOR DYEING MATERIALS CONTAINING HYDROXYL OR AMIDE GROUPS BAYER AG (DE) 1982-09-15 EP disclosed
EP-0013879-A1 Reactive dyestuffs, their preparation and their use for dyeing materials containing hydroxyl or amide groups BAYER AG (DE) 1980-08-06 EP disclosed
US-4052212-A ETHER-ESTER KONISHIROKU PHOTO INDUSTRY CO., LTD. (JA) 1977-10-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100152190-A1 Substituted Pyrrolidine-2-Carboxamides ARG2, CCNY, PYCR1 LMNA 3002/4885CYP1A2 730/4885CYP3A4 740/4885
US-20100075948-A1 Substituted Pyrrolidine-2-Carboxamides ARG2, CCNY, PYCR1 LMNA 3002/4885CYP1A2 730/4885CYP3A4 740/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.