SCHEMBL3377149

SCHEMBL3377149

O=C(O)OCc1cc(-c2cccc(Cl)c2)c2nccn2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.43
EPHB4 P54760 3/20 0.41
GPR119 Q8TDV5 1/20 0.41
XDH P47989 1/20 0.39
SLC22A12 Q96S37 1/20 0.39
RET P07949 1/20 0.38
PTGER1 P34995 2/20 0.38
EGLN1 Q9GZT9 1/20 0.38
NAMPT P43490 1/20 0.38
SPTLC1 O15269 1/20 0.37
JAK2 O60674 3/20 0.37
CYP3A4 P08684 1/20 0.37
FFAR1 O14842 2/20 0.36
KMO O15229 1/20 0.36
HCAR2 Q8TDS4 1/20 0.36
ABL1 P00519 1/20 0.36
EGFR P00533 1/20 0.36
SRC P12931 1/20 0.36
KDR P35968 1/20 0.36
ABL2 P42684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7913069 0.89 HDAC6 (0.44) HDAC6EPHB4GPR119RETNAMPT
SCHEMBL3380305 0.83 HDAC6 (0.44) HDAC6EPHB4XDHSLC22A12RET
SCHEMBL3377436 0.76 HDAC6 (0.39) HDAC6EPHB4RETNAMPTCYP3A4
SCHEMBL3379666 0.76 MAPK14 (0.48) HDAC6EPHB4SPTLC1JAK2CYP3A4
SCHEMBL7911311 0.73 HDAC6 (0.37) HDAC6EPHB4RETNAMPTJAK2
SCHEMBL3379763 0.72 TRPM8 (0.39) GPR119EGFR
SCHEMBL21439356 0.70 CFD (0.65) PTGER1
SCHEMBL21439496 0.70 HDAC6 (0.43) HDAC6EPHB4XDHSLC22A12NAMPT
SCHEMBL3381843 0.69 GPR119 (0.39) GPR119EGLN1JAK2EGFR
SCHEMBL11920620 0.67 IKBKB (0.39) FFAR1HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059838-A2 PDE4 INHIBITORS SELECTIVE FOR THE LONG FORM OF PDE4 FOR TREATING INFLAMMATION AND AVOIDING SIDE EFFECTS DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed