SCHEMBL3377436

SCHEMBL3377436

Nc1ccc(Cc2cc(-c3cccc(Cl)c3)c3nccn3c2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.39
KDR P35968 2/20 0.37
ABL1 P00519 1/20 0.37
EGFR P00533 1/20 0.37
SRC P12931 1/20 0.37
ABL2 P42684 1/20 0.37
DHFR P00374 1/20 0.37
PDE4D Q08499 1/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
MAOB P27338 2/20 0.36
EPHB4 P54760 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
MAP4K4 O95819 1/20 0.36
RET P07949 1/20 0.35
TDO2 P48775 1/20 0.35
CYP17A1 P05093 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7911311 0.84 HDAC6 (0.37) HDAC6KDRDHFRNPC1RAB9A
SCHEMBL3380305 0.82 HDAC6 (0.44) HDAC6KDRNPC1RAB9AMEN1
SCHEMBL7905671 0.81 PDE4D (0.39) KDRABL1EGFRSRCABL2
SCHEMBL3428353 0.78 RAB9A (0.40) KDRABL1EGFRSRCABL2
SCHEMBL3433258 0.76 DPP4 (0.38) KDRABL1EGFRSRCABL2
SCHEMBL3377149 0.76 HDAC6 (0.43) HDAC6KDRABL1EGFRSRC
SCHEMBL7913069 0.73 HDAC6 (0.44) HDAC6EGFRPDE4DEPHB4RET
SCHEMBL14006703 0.72 HDAC6 (0.50) HDAC6KDRABL1EGFRSRC
SCHEMBL3378478 0.71 DHFR (0.39) KDRABL1EGFRSRCABL2
SCHEMBL16114143 0.70 PDE4D (0.47) DHFRPDE4DMAOBTAAR1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059838-A2 PDE4 INHIBITORS SELECTIVE FOR THE LONG FORM OF PDE4 FOR TREATING INFLAMMATION AND AVOIDING SIDE EFFECTS DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed
WO-2010059838-A2 PDE4 INHIBITORS SELECTIVE FOR THE LONG FORM OF PDE4 FOR TREATING INFLAMMATION AND AVOIDING SIDE EFFECTS DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed