Gf-109203

Gf-109203

SCHEMBL338086

CN(C)CCCn1cc(C2=C(c3c[nH]c4ccccc34)C(=O)NC2=O)c2ccccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKACA P17612 13/20 1.00
PRKACG P22612 13/20 1.00
PRKACB P22694 13/20 1.00
PRKCA P17252 5/20 1.00
CDK4 P11802 4/20 1.00
CCND1 P24385 4/20 1.00
PRKCB P05771 4/20 1.00
PRKCH P24723 3/20 1.00
PRKCQ Q04759 3/20 1.00
PRKCD Q05655 3/20 1.00
PRKCE Q02156 3/20 1.00
CCNB2 O95067 3/20 1.00
CDK1 P06493 3/20 1.00
CCNB1 P14635 3/20 1.00
CCNB3 Q8WWL7 3/20 1.00
PRKD1 Q15139 2/20 1.00
TDP1 Q9NUW8 2/20 1.00
PIM1 P11309 2/20 1.00
GSK3B P49841 2/20 1.00
CCNE2 O96020 2/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Gf-109203 SCHEMBL29353725 1.00 PRKACA (1.00) PRKACAPRKACGPRKACBPRKCACDK4
Gf-109203 SCHEMBL29534077 0.99 PRKACA (0.98) PRKACAPRKACGPRKACBPRKCACDK4
Gf-109203 SCHEMBL1199513 0.99 PRKACA (0.98) PRKACAPRKACGPRKACBPRKCACDK4
SCHEMBL7823516 0.94 PRKACA (0.88) PRKACAPRKACGPRKACBPRKCACDK4
SCHEMBL14022587 0.92 PRKACA (0.85) PRKACAPRKACGPRKACBPRKCACDK4
SCHEMBL9086320 0.90 PRKACA (0.82) PRKACAPRKACGPRKACBPRKCACDK4
SCHEMBL9087076 0.90 PRKACA (0.82) PRKACAPRKACGPRKACBPRKCACDK4
SCHEMBL9087451 0.90 PRKACA (0.82) PRKACAPRKACGPRKACBPRKCACDK4
SCHEMBL7826095 0.90 PRKACA (0.81) PRKACAPRKACGPRKACBPRKCACDK4
SCHEMBL7815621 0.90 PRKACA (0.81) PRKACAPRKACGPRKACBPRKCACDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 304 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2797596-B1 PERITONEAL DIALYSIS FLUID COMPRISING A GSK-3 INHIBITOR ZYTOPROTEC GMBH (AT) 2019-06-26 EP claimed
US-20150004255-A1 PERITONEAL DIALYSIS FLUID COMPRISING A GSK-3 INHIBITOR ZYTOPROTEC GMBH (AT) 2015-01-01 US claimed
CN-104023722-A Peritoneal dialysis fluid comprising GSK-3 inhibitor ZYTOPROTEC GMBH 2014-09-03 CN claimed
WO-2014081922-A1 COMPOSITIONS AND METHODS USEFUL IN PREVENTING AND TREATING APICOMPLEXA INFECTIONS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2014-05-30 WO claimed
EP-2653166-A2 Pharmaceutical composition and related methods Healor Ltd. (IL) 2013-10-23 EP claimed
EP-2609918-A1 Peritoneal dialysis fluid comprising a GSK-3 inhibitor Zytoprotec GmbH (AT) 2013-07-03 EP claimed
CN-102755649-A Pharmaceutical composition and related methods HEALOR LTD 2012-10-31 CN claimed
US-20120238019-A1 STEM CELL CULTURE MEDIA FOR MAINTAINING STEMNESS OR INDUCING DIFFERENTIATION OF STEM CELLS COLLEGE OF MEDICINE POCHON CHA UNIVERSITY INDUSTRY-ACADEMIC COOPERATION FOUNDATION (KR) 2012-09-20 US claimed
EP-2494865-A2 GUT FLORA-DERIVED EXTRACELLULAR VESICLES, AND METHOD FOR SEARCHING FOR A DISEASE MODEL, VACCINE, AND CANDIDATE DRUG AND FOR DIAGNOSIS USING SAME Aeon Medix Inc. (KR) 2012-09-05 EP claimed
US-20100310542-A1 Pharmaceutical Compositions for treating wouds and related methods HEALOR LTD. (IL) 2010-12-09 US claimed
EP-2185184-A2 PHARMACEUTICAL COMPOSITION FOR TREATING WOUNDS AND RELATED METHODS HealOr Ltd. (IL) 2010-05-19 EP claimed
WO-2009016629-A2 PHARMACEUTICAL COMPOSITION FOR TREATING WOUNDS AND RELATED METHODS HEALOR LTD. (IL) 2009-02-05 WO claimed
US-20080009511-A1 Cancer treatment with compounds inhibiting PKC alpha LU ZHIMIN 2008-01-10 US claimed
US-20070196514-A1 Prostate cancer treatment with glycogen synthase kinase-3beta inhibitors UNIVERSITY OF KANSAS MEDICAL CENTER 2007-08-23 US claimed
US-20060099568-A1 Signals and molecular species involved in senescence SEOUL NATIONAL UNIVERSITY INDUSTRY FOUNDATION (KR) 2006-05-11 US claimed
US-20060009492-A1 Cancer treatment with compounds inhibiting PKC alpha LU ZHIMIN 2006-01-12 US claimed
WO-2003104482-A1 SIGNALS AND MOLECULAR SPECIES INVOLVED IN SENESCENCE METABOLIC ENGINEERING LABORATORIES CO., LTD. (KR) 2003-12-18 WO claimed
EP-0397060-B1 Maleinimide derivatives and their use as medicines GOEDECKE AG (DE) 2001-11-21 EP claimed
EP-4678737-A1 METHOD FOR PRODUCING PRIMED PLURIPOTENT STEM CELLS Kyoto University (JP) 2026-01-14 EP disclosed
US-5380746-A Bis-(1H-indol-3-YL)-maleinimide derivatives, processes for the preparation thereof and pharmaceutical compositions containing them GOEDECKE AKTIENGESELLSCHAFT (DE) 1995-01-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100310542-A1 Pharmaceutical Compositions for treating wouds and related methods PRKCZ, PRKCB, PRKCA PRKACA 9/4885PRKACG 15/4885PRKACB 14/4885
US-20080009511-A1 Cancer treatment with compounds inhibiting PKC alpha PRKCE, ROCK1, PRKCA PRKACA 15/4885PRKACG 36/4885PRKACB 32/4885
US-20060009492-A1 Cancer treatment with compounds inhibiting PKC alpha PRKCE, ROCK1, PRKCA PRKACA 15/4885PRKACG 36/4885PRKACB 32/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.