SCHEMBL338573

SCHEMBL338573

N#Cc1cc2nccn2cc1Br

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.41
PDE3A Q14432 1/20 0.41
CYP3A4 P08684 1/20 0.40
HPGD P15428 1/20 0.40
NFKB1 P19838 1/20 0.40
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40
HSD17B10 Q99714 1/20 0.40
DYRK1A Q13627 2/20 0.34
KEAP1 Q14145 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
AXL P30530 1/20 0.34
FLT3 P36888 1/20 0.34
MERTK Q12866 1/20 0.34
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
KMT2A Q03164 1/20 0.33
TRIM33 Q9UPN9 1/20 0.32
GRM4 Q14833 1/20 0.31
ABL1 P00519 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL407441 0.77 L3MBTL1 (0.49) PDE4APDE3ACYP3A4HPGDNFKB1
SCHEMBL24087299 0.76 PDE4A (0.41) PDE4APDE3ACYP3A4HPGDNFKB1
SCHEMBL12618998 0.76 PDE4A (0.47) PDE4APDE3ACYP3A4HPGDNFKB1
SCHEMBL30446178 0.76 PDE4A (0.41) PDE4APDE3ACYP3A4HPGDNFKB1
Hydrochloric Acid SCHEMBL31647268 0.75 L3MBTL1 (0.47) PDE4APDE3ACYP3A4HPGDNFKB1
SCHEMBL25233154 0.73 DYRK1A (0.41) DYRK1AKEAP1L3MBTL1AXLMEN1
SCHEMBL24087352 0.73 TGFBR1 (0.38) DYRK1AKEAP1L3MBTL1MEN1CYP1A2
SCHEMBL21646478 0.72 PDE4A (0.41) PDE4APDE3ACYP3A4HPGDNFKB1
SCHEMBL25104400 0.71 GRM5 (0.34) L3MBTL1MEN1KMT2A
SCHEMBL339104 0.69 KDM4E (0.45) PDE4APDE3ACYP3A4HPGDNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230303569-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS ARISAN THERAPEUTICS INC. (US) 2023-09-28 US disclosed
US-20230303569-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS ARISAN THERAPEUTICS INC. (US) 2023-09-28 US disclosed
US-20230303569-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS ARISAN THERAPEUTICS INC. (US) 2023-09-28 US disclosed
US-20220193038-A1 COMPOUNDS FOR THE TREATMENT OF ARENAVIRUS INFECTION ARISAN THERAPEUTICS INC. (US) 2022-06-23 US disclosed
WO-2022108849-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS ARISAN THERAPEUTICS INC. (US) 2022-05-27 WO disclosed
WO-2022108849-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS ARISAN THERAPEUTICS INC. (US) 2022-05-27 WO disclosed
EP-3890731-A1 COMPOUNDS FOR THE TREATMENT OF ARENAVIRUS INFECTION Arisan Therapeutics, Inc. (US) 2021-10-13 EP disclosed
CN-113329750-A Compounds for the treatment of arenavirus infections 阿里桑治疗药物公司 2021-08-31 CN disclosed
WO-2020117794-A1 COMPOUNDS FOR THE TREATMENT OF ARENAVIRUS INFECTION ARISAN THERAPEUTICS, INC. (US) 2020-06-11 WO disclosed
WO-2020117794-A1 COMPOUNDS FOR THE TREATMENT OF ARENAVIRUS INFECTION ARISAN THERAPEUTICS, INC. (US) 2020-06-11 WO disclosed
US-20120077787-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2012-03-29 US disclosed
US-20120077787-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2012-03-29 US disclosed
US-8097617-B2 Organic compounds NOVARTIS AG (CH) 2012-01-17 US disclosed
US-8097617-B2 Organic compounds NOVARTIS AG (CH) 2012-01-17 US disclosed
US-20090253689-A1 Organic Compounds NOVARTIS AG (CH) 2009-10-08 US disclosed
US-20090253689-A1 Organic Compounds NOVARTIS AG (CH) 2009-10-08 US disclosed
EP-2004643-A1 ORGANIC COMPOUNDS Novartis AG (CH) 2008-12-24 EP disclosed
WO-2007113226-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2007-10-11 WO disclosed
WO-2007113226-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2007-10-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120077787-A1 ORGANIC COMPOUNDS OAT, GPR119, OTC PDE4A 3042/4885PDE3A 1335/4885CYP3A4 85/4885
US-20220193038-A1 COMPOUNDS FOR THE TREATMENT OF ARENAVIRUS INFECTION HAVCR2, ZC3HAV1, CD4 PDE4A 3068/4885PDE3A 4166/4885CYP3A4 2120/4885
US-20230303569-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS C3AR1, C9, C1R PDE4A 3997/4885PDE3A 3201/4885CYP3A4 344/4885
US-20090253689-A1 Organic Compounds OAT, GPR119, OTC PDE4A 3042/4885PDE3A 1335/4885CYP3A4 85/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.