SCHEMBL3386876

SCHEMBL3386876

O=C(c1ccc2[nH]ccc2c1)N1CCN(C2CCCC2)CC1.O=C(c1ccc2c(ccn2C[C@@H]2CCCN2Cc2ccccc2)c1)N1CCN(C2CCCC2)CC1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.54
CCR3 P51677 1/20 0.46
CHRM2 P08172 1/20 0.44
OXTR P30559 3/20 0.43
ACHE P22303 2/20 0.42
HTR4 Q13639 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 3/20 0.41
KMT2A Q03164 1/20 0.41
POLB P06746 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ACACB O00763 1/20 0.41
ACACA Q13085 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3383896 0.92 OXTR (0.48) OXTRACHEKDM4EALDH1A1KMT2A
SCHEMBL3387941 0.89 MAPK14 (0.53) MAPK14CCR3CHRM2OXTRACHE
SCHEMBL3387677 0.87 MAPK14 (0.56) MAPK14CCR3CHRM2ACHEHTR4
SCHEMBL3388485 0.85 MAPK14 (0.56) MAPK14CCR3CHRM2ACHEHTR4
SCHEMBL3383892 0.82 MAPK14 (0.64) MAPK14CCR3CHRM2ACHEHTR4
SCHEMBL3943261 0.81 HRH3 (0.57) ACHEKDM4EALDH1A1KMT2APOLB
SCHEMBL3390277 0.80 MAPK14 (0.60) MAPK14CCR3CHRM2OXTRACHE
SCHEMBL3387892 0.80 OXTR (0.47) OXTRACHEKDM4EHRH3
SCHEMBL3388617 0.80 DRD2 (0.52) MAPK14CCR3CHRM2KDM4EALDH1A1
SCHEMBL3388657 0.79 MAPK14 (0.60) MAPK14CCR3CHRM2OXTRACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029534-B1 1H-INDOL-5-YL-PIPERAZIN-1-YL-METHANONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2010-12-22 EP disclosed