SCHEMBL3392203

SCHEMBL3392203

FC(F)(F)Oc1ccc(CNCCc2cc3cc(Br)ccc3s2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN8A Q9UQD0 1/20 0.40
HDAC6 Q9UBN7 1/20 0.38
USP28 Q96RU2 1/20 0.37
USP25 Q9UHP3 1/20 0.37
HDAC1 Q13547 1/20 0.36
HTR2A P28223 3/20 0.35
KCNN3 Q9UGI6 1/20 0.35
CHEK1 O14757 1/20 0.34
HSP90AA1 P07900 1/20 0.33
GPR39 O43194 1/20 0.33
SLC6A5 Q9Y345 1/20 0.33
PPARA Q07869 1/20 0.33
WDR5 P61964 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA9 Q16790 1/20 0.33
LTA4H P09960 1/20 0.33
EPHX2 P34913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3392201 0.76 SLC6A4 (0.38) HDAC6HSP90AA1
SCHEMBL3392210 0.70 PRMT1 (0.47) SCN8AHTR2ACHEK1CA12CA1
SCHEMBL15984865 0.70 TAAR1 (0.44) CHEK1HSP90AA1
SCHEMBL8348550 0.68 SCN8A (0.55) SCN8AEPHX2
SCHEMBL4575327 0.68 BCHE (0.59) SCN8ASLC6A5CA1CA2LTA4H
SCHEMBL3396182 0.67 CLK1 (0.57) HDAC6HDAC1PPARA
Hydrochloric Acid SCHEMBL6122751 0.67 SCN8A (0.54) SCN8AEPHX2
SCHEMBL15980807 0.67 LMNA (0.39) HSP90AA1PPARA
SCHEMBL19243611 0.66 SCN8A (0.55) SCN8AHDAC6HDAC1EPHX2
SCHEMBL9903315 0.66 SCN8A (0.58) SCN8ASLC6A5CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2246329-A1 4(1H)-pyridinone derivatives and their use as antimalaria agents Glaxo Group Limited (GB) 2010-11-03 EP disclosed