SCHEMBL3393091

SCHEMBL3393091

C#CCN(C)Cc1ccc(OC(F)(F)F)cc1

nearest known ligand 0.67

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 18/20 0.67
MAOB P27338 2/20 0.57
LMNA P02545 2/20 0.56
USP2 O75604 1/20 0.56
CYP3A4 P08684 1/20 0.56
TSHR P16473 1/20 0.56
MAOA P21397 1/20 0.56
ALDH1A1 P00352 1/20 0.54
BLM P54132 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
SLC6A4 P31645 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3393368 0.85 PYCR1 (0.59) PYCR1MAOBTSHRALDH1A1SLC6A4
SCHEMBL3396909 0.85 SLC6A4 (0.56) PYCR1MAOBMAOAALDH1A1SLC6A4
SCHEMBL13074386 0.85 SLC6A4 (0.57) PYCR1TSHRALDH1A1SLC6A4
SCHEMBL3394463 0.81 PYCR1 (0.47) PYCR1MAOBTSHRMAOASLC6A4
SCHEMBL3394172 0.79 PYCR1 (1.00) PYCR1MAOBLMNAUSP2CYP3A4
SCHEMBL8244727 0.78 PYCR1 (0.72) PYCR1MAOBLMNAUSP2CYP3A4
SCHEMBL2056224 0.78 SLC6A4 (0.66) TSHRALDH1A1SLC6A4
SCHEMBL13070308 0.78 PRMT6 (0.51) TSHRALDH1A1SLC6A4
SCHEMBL3423840 0.78 SLC6A4 (0.50) PYCR1MAOBTSHRALDH1A1SLC6A4
SCHEMBL13070333 0.78 SLC6A4 (0.50) PYCR1MAOBTSHRALDH1A1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2246329-A1 4(1H)-pyridinone derivatives and their use as antimalaria agents Glaxo Group Limited (GB) 2010-11-03 EP disclosed