SCHEMBL3394463

SCHEMBL3394463

C#CCN(CCC)Cc1ccc(OC(F)(F)F)cc1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 4/20 0.47
HRH3 Q9Y5N1 1/20 0.44
TSHR P16473 1/20 0.43
SLC6A4 P31645 3/20 0.42
SLC6A3 Q01959 2/20 0.41
MAOB P27338 5/20 0.41
MAOA P21397 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3393091 0.81 PYCR1 (0.67) PYCR1TSHRSLC6A4MAOBMAOA
SCHEMBL12963728 0.78 TSHR (0.53) HRH3TSHRSLC6A4SLC6A3
SCHEMBL13070308 0.77 PRMT6 (0.51) TSHRSLC6A4SLC6A3
SCHEMBL3393368 0.75 PYCR1 (0.59) PYCR1TSHRSLC6A4SLC6A3MAOB
SCHEMBL3396909 0.75 SLC6A4 (0.56) PYCR1SLC6A4SLC6A3MAOBMAOA
SCHEMBL27210386 0.75 PYCR1 (0.72) PYCR1MAOBMAOA
SCHEMBL17914547 0.74 TSHR (0.46) HRH3TSHRSLC6A4SLC6A3
SCHEMBL14376823 0.74 SLC6A4 (0.50) HRH3TSHRSLC6A4SLC6A3
SCHEMBL3397214 0.73 PYCR1 (0.41) PYCR1TSHRSLC6A4
SCHEMBL14376814 0.72 SLC6A4 (0.48) TSHRSLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2246329-A1 4(1H)-pyridinone derivatives and their use as antimalaria agents Glaxo Group Limited (GB) 2010-11-03 EP disclosed