SCHEMBL3396909

SCHEMBL3396909

C#CCN(C)CCc1ccc(OC(F)(F)F)cc1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.56
SLC6A3 Q01959 4/20 0.56
PYCR1 P32322 6/20 0.48
MAOB P27338 2/20 0.46
MAOA P21397 1/20 0.46
ACHE P22303 2/20 0.45
ALDH1A1 P00352 1/20 0.41
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3393091 0.85 PYCR1 (0.67) SLC6A4PYCR1MAOBMAOAALDH1A1
SCHEMBL5667997 0.79 SLC6A4 (0.58) SLC6A4SLC6A3ALDH1A1
Hydrochloric Acid SCHEMBL8508484 0.78 SLC6A4 (0.57) SLC6A4SLC6A3ALDH1A1
SCHEMBL3393368 0.77 PYCR1 (0.59) SLC6A4SLC6A3PYCR1MAOBACHE
SCHEMBL3394463 0.75 PYCR1 (0.47) SLC6A4SLC6A3PYCR1MAOBMAOA
SCHEMBL1176965 0.74 MAOA (0.67) PYCR1MAOBMAOAACHEALDH1A1
Hydrochloric Acid SCHEMBL28077090 0.73 LMNA (0.68) PYCR1MAOBMAOAACHEALDH1A1
SCHEMBL13074386 0.72 SLC6A4 (0.57) SLC6A4SLC6A3PYCR1ACHEALDH1A1
SCHEMBL3215494 0.72 ALDH1A1 (0.44) SLC6A4ACHEALDH1A1
SCHEMBL1971365 0.72 SLC6A4 (0.54) SLC6A4SLC6A3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2246329-A1 4(1H)-pyridinone derivatives and their use as antimalaria agents Glaxo Group Limited (GB) 2010-11-03 EP disclosed
WO-2010081904-A1 4 ( 1H) -PYRIDINONE DERIVATIVES AND THEIR USE AS ANTIMALARIA AGENTS GLAXO GROUP LIMITED (GB) 2010-07-22 WO disclosed