SCHEMBL3393224

SCHEMBL3393224

Cc1ccc(-n2nc(C(C)(C)C)cc2N(OS(C)(=O)=O)C(=O)Nc2ccc(N3CCN(C(=O)c4ccccc4Cl)CC3)nc2C)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.38
KDM4E B2RXH2 4/20 0.37
GAA P10253 2/20 0.37
ALDH1A1 P00352 2/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PTK2B Q14289 1/20 0.36
KMT2A Q03164 2/20 0.36
MAPK14 Q16539 4/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
ALOX12 P18054 1/20 0.35
JAK2 O60674 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
DCTPP1 Q9H773 1/20 0.34
MAPK13 O15264 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3391158 0.93 GBA1 (0.37) GBA1KDM4EGAAALDH1A1HTT
SCHEMBL3393213 0.93 PTK2B (0.38) KDM4ESMN1; SMN2PTK2BMAPK14HSD17B10
SCHEMBL3389419 0.92 ALDH1A1 (0.39) KDM4EGAAALDH1A1PTK2BKMT2A
SCHEMBL3393250 0.92 MAPK12 (0.40) GBA1KDM4EGAAALDH1A1HTT
SCHEMBL3391110 0.91 GBA1 (0.41) GBA1DCTPP1
SCHEMBL3389769 0.90 JAK2 (0.37) KDM4EGAAALDH1A1HTTSMN1; SMN2
SCHEMBL3394251 0.90 PTK2B (0.39) GBA1KDM4EALDH1A1HTTSMN1; SMN2
SCHEMBL3422290 0.90 MAPK14 (0.37) GBA1KDM4EGAAALDH1A1HTT
SCHEMBL3392554 0.89 PTK2B (0.37) KDM4EALDH1A1HTTSMN1; SMN2PTK2B
SCHEMBL3392100 0.89 PTK2B (0.39) PTK2BKMT2AMAPK14LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943243-B1 KINASE INHIBITORS LILLY CO ELI (US) 2010-12-29 EP disclosed