SCHEMBL3393472

SCHEMBL3393472

C#CCN1CCC(c2ccc(OC(F)(F)F)cc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOB P27338 13/20 0.50
MAOA P21397 5/20 0.50
MMP1 P03956 1/20 0.44
MMP13 P45452 1/20 0.44
MMP14 P50281 1/20 0.44
P2RY14 Q15391 1/20 0.43
EPHX2 P34913 1/20 0.43
DRD2 P14416 1/20 0.43
FAAH O00519 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19538689 0.81 TSHR (0.60) EPHX2DRD2FAAH
SCHEMBL4564168 0.77 L3MBTL1 (0.47) EPHX2FAAH
SCHEMBL14438091 0.76 HTR2A (0.53) MAOBEPHX2DRD2FAAH
SCHEMBL81671 0.76 MAOB (0.60) MAOBMAOADRD2
SCHEMBL3392222 0.76 MAOA (0.58) MAOBMAOADRD2
SCHEMBL22816265 0.75 EPHX2 (0.38) EPHX2FAAH
SCHEMBL3398473 0.75 TEAD1 (0.57) DRD2
SCHEMBL3392273 0.75 FAAH (0.39) EPHX2DRD2FAAH
SCHEMBL28247613 0.73 MEN1 (0.48) EPHX2FAAH
SCHEMBL64479 0.73 MAOB (0.48) MAOBMAOAP2RY14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2246329-A1 4(1H)-pyridinone derivatives and their use as antimalaria agents Glaxo Group Limited (GB) 2010-11-03 EP disclosed