SCHEMBL3392222

SCHEMBL3392222

C#CCN1CCC(c2ccccc2)CC1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOA P21397 6/20 0.58
MAOB P27338 5/20 0.58
SLC18A3 Q16572 3/20 0.57
DRD2 P14416 1/20 0.57
SIGMAR1 Q99720 4/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
CARM1 Q86X55 1/20 0.53
PRMT6 Q96LA8 1/20 0.53
TP53 P04637 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
TSHR P16473 1/20 0.51
CYP2C19 P33261 1/20 0.51
BCHE P06276 1/20 0.50
KCNA3 P22001 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL81671 0.83 MAOB (0.60) MAOAMAOBSLC18A3DRD2
SCHEMBL9476556 0.83 SLC18A3 (0.63) SLC18A3DRD2SIGMAR1MEN1KMT2A
SCHEMBL14328412 0.82 SLC18A3 (0.57) SLC18A3DRD2SIGMAR1MEN1KMT2A
SCHEMBL10696270 0.82 SLC18A3 (0.57) SLC18A3DRD2SIGMAR1MEN1KMT2A
SCHEMBL16364107 0.81 DRD2 (0.67) MAOAMAOBDRD2BCHE
SCHEMBL16829624 0.81 DRD2 (0.63) MAOBDRD2SIGMAR1
SCHEMBL22485567 0.79 DRD2 (0.58) SLC18A3DRD2SIGMAR1MEN1KMT2A
SCHEMBL7403433 0.77 MAOB (0.49) MAOAMAOBBCHE
SCHEMBL9369758 0.76 SLC18A3 (0.69) SLC18A3DRD2SIGMAR1MEN1KMT2A
SCHEMBL18026661 0.76 MAOA (0.72) MAOAMAOBSIGMAR1CARM1PRMT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0537008-B1 Use of biphosphonates for the manufacture of a medicament for blocking neoplastic transformation of cells induced by ras oncogenes SQUIBB & SONS INC (US) 1995-10-25 EP claimed
US-20260125349-A1 PROCESS FOR THE FLUORINATION AND/OR CYCLIZATION OF AN AMINO ALKENE OR ALKYNE IN A CONTINUOUS STREAM AND FACILITY FOR PERFORMING THE PROCESS UNIV POITIERS (FR) 2026-05-07 US disclosed
EP-4598903-A1 PROCESS FOR THE FLUORINATION AND/OR CYCLIZATION OF AN AMINO ALKENE OR ALKYNE IN A CONTINUOUS STREAM AND FACILITY FOR PERFORMING THE PROCESS Université de Poitiers (FR) 2025-08-13 EP disclosed
CN-120035579-A Process for fluorinating and/or cyclizing an amino alkene or alkyne in a continuous flow and apparatus for carrying out the process 普瓦捷大学 2025-05-23 CN disclosed
WO-2024074501-A1 PROCESS FOR THE FLUORINATION AND/OR CYCLIZATION OF AN AMINO ALKENE OR ALKYNE IN A CONTINUOUS STREAM AND FACILITY FOR PERFORMING THE PROCESS UNIVERSITE DE POITIERS (FR) 2024-04-11 WO disclosed
US-10301267-B2 Compounds ASTRAZENECA AB (SE) 2019-05-28 US disclosed
US-9902711-B2 Piperidine compounds having multimodal activity against pain LABORATORIOS DEL DR. ESTEVE S.A. (ES) 2018-02-27 US disclosed
US-20170260143-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2017-09-14 US disclosed
US-9688640-B2 Methods of treating cancer with a pyrazole derivative ASTRAZENECA AB (SE) 2017-06-27 US disclosed
US-20170001979-A1 Piperidine compounds having multimodal activity against pain ESTEVE PHARMACEUTICALS, S.A. (ES) 2017-01-05 US disclosed
EP-2246329-A1 4(1H)-pyridinone derivatives and their use as antimalaria agents Glaxo Group Limited (GB) 2010-11-03 EP disclosed
WO-2010081904-A1 4 ( 1H) -PYRIDINONE DERIVATIVES AND THEIR USE AS ANTIMALARIA AGENTS GLAXO GROUP LIMITED (GB) 2010-07-22 WO disclosed
EP-1423363-B1 ORAL ANTIDIABETIC AGENTS WARNER LAMBERT CO (US) 2006-04-19 EP disclosed
EP-1577305-A1 Oral antidiabetic agents WARNER-LAMBERT COMPANY LLC (US) 2005-09-21 EP disclosed
CN-1558897-A oral antidiabetic agent ����-�����ع�˾ 2004-12-29 CN disclosed
EP-1423363-A1 ORAL ANTIDIABETIC AGENTS Warner-Lambert Company LLC (US) 2004-06-02 EP disclosed
US-20030171377-A1 Antidiabetic agents BIGGE CHRISTOPHER FRANKLIN (US) 2003-09-11 US disclosed
WO-2003018553-A1 ORAL ANTIDIABETIC AGENTS WARNER-LAMBERT COMPANY LLC (US) 2003-03-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030171377-A1 Antidiabetic agents SLC5A1, SLC5A2, GLP1R MAOA 1046/4885MAOB 316/4885SLC18A3 3547/4885
US-10301267-B2 Compounds SLC10A1, CYP11B1, ABCB11 MAOA 1555/4885MAOB 1283/4885SLC18A3 3899/4885
US-20260125349-A1 PROCESS FOR THE FLUORINATION AND/OR CYCLIZATION OF AN AMINO ALKENE OR ALKYNE IN A CONTINUOUS STREAM AND FACILITY FOR PERFORMING THE PROCESS FIBP, FGB, SUB1 MAOA 876/4885MAOB 343/4885SLC18A3 3536/4885
US-20170260143-A1 NOVEL COMPOUNDS SLC10A1, ABCB11, CYP11B1 MAOA 3474/4885MAOB 2776/4885SLC18A3 3829/4885
US-20170001979-A1 Piperidine compounds having multimodal activity against pain OPRD1, OPRM1, OPRL1 MAOA 947/4885MAOB 1266/4885SLC18A3 934/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.