SCHEMBL3396747

SCHEMBL3396747

CCn1cc(CN2CCC(N3CCCC3)CC2)nc1-c1cccc2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
RECQL P46063 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MBTD1 Q05BQ5 1/20 0.40
L3MBTL3 Q96JM7 1/20 0.40
HRH3 Q9Y5N1 1/20 0.39
ACHE P22303 1/20 0.39
TACR2 P21452 4/20 0.39
TACR3 P29371 4/20 0.39
OPRM1 P35372 3/20 0.39
TRPV4 Q9HBA0 7/20 0.38
OPRK1 P41145 1/20 0.37
OPRL1 P41146 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3399916 0.99 ALDH1A1 (0.42) ALDH1A1TSHRRECQLL3MBTL1MBTD1
SCHEMBL13310392 0.99 ALDH1A1 (0.42) ALDH1A1TSHRRECQLL3MBTL1MBTD1
SCHEMBL3404354 0.92 SIGMAR1 (0.46) ALDH1A1ACHETACR2TACR3OPRM1
SCHEMBL3399827 0.92 SIGMAR1 (0.43) ALDH1A1HRH3ACHETACR2TACR3
SCHEMBL3399762 0.84 KMT2A (0.45) ALDH1A1
SCHEMBL3396799 0.84 ACHE (0.40) ALDH1A1ACHE
SCHEMBL3404844 0.80 ACHE (0.36) TSHRACHE
SCHEMBL3402347 0.79 LMNA (0.36) ALDH1A1ACHETACR2TACR3OPRM1
SCHEMBL3402431 0.79 CCND1 (0.40) ACHETACR2TACR3OPRM1
SCHEMBL3405131 0.79 TLR8 (0.43) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed