SCHEMBL3400542

SCHEMBL3400542

COc1ccc(CO[C@@H]2C[C@H](CC=O)N(C(=O)OCc3ccccc3)C2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.45
BDKRB2 P30411 2/20 0.45
ALDH1A1 P00352 1/20 0.44
NPSR1 Q6W5P4 1/20 0.43
TP53 P04637 1/20 0.43
ITGB3 P05106 3/20 0.42
ITGB1 P05556 3/20 0.42
ITGAV P06756 3/20 0.42
ITGA5 P08648 3/20 0.42
ITGB5 P18084 3/20 0.42
P2RX4 Q99571 1/20 0.42
ITGA2B P08514 2/20 0.41
MMP1 P03956 1/20 0.41
MMP3 P08254 1/20 0.41
MMP7 P09237 1/20 0.41
MMP9 P14780 1/20 0.41
MMP13 P45452 1/20 0.41
PARP1 P09874 1/20 0.40
CHRM5 P08912 1/20 0.40
CHRM1 P11229 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL115938 1.00 ABCB1 (0.45) ABCB1BDKRB2ALDH1A1NPSR1TP53
SCHEMBL178628 0.91 ABCB1 (0.44) ABCB1BDKRB2ALDH1A1NPSR1TP53
SCHEMBL116032 0.89 BDKRB2 (0.47) ABCB1BDKRB2ALDH1A1NPSR1TP53
SCHEMBL13625886 0.87 BDKRB2 (0.52) ABCB1BDKRB2ALDH1A1CHRM5CHRM1
SCHEMBL116901 0.87 BDKRB2 (0.46) ABCB1BDKRB2ALDH1A1NPSR1TP53
SCHEMBL3398953 0.87 ALDH1A1 (0.46) BDKRB2ALDH1A1NPSR1TP53P2RX4
SCHEMBL116053 0.87 ALDH1A1 (0.46) BDKRB2ALDH1A1NPSR1TP53P2RX4
SCHEMBL114544 0.86 BDKRB2 (0.45) ABCB1BDKRB2ALDH1A1NPSR1TP53
SCHEMBL116041 0.83 AGTR2 (0.48) BDKRB2ALDH1A1NPSR1TP53P2RX4
SCHEMBL3402980 0.83 ALDH1A1 (0.44) BDKRB2ALDH1A1NPSR1TP53P2RX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250171-A2 ANTIBACTERIAL FLUOROQUINOLONE ANALOGS Achaogen, Inc. (US) 2010-11-17 EP disclosed
WO-2009137130-A2 ANTIBACTERIAL FLUOROQUINOLONE ANALOGS ACHAOGEN, INC. (US) 2009-11-12 WO disclosed