SCHEMBL340107

SCHEMBL340107

O=C(Cl)c1cccc(OCc2ccccc2)c1

nearest known ligand 0.77

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 6/20 0.77
MAOB P27338 3/20 0.72
SMPD1 P17405 2/20 0.68
SRD5A2 P31213 1/20 0.67
PTPN1 P18031 1/20 0.65
MEN1 O00255 1/20 0.61
KMT2A Q03164 1/20 0.61
NR1H4 Q96RI1 1/20 0.59
MAOA P21397 2/20 0.58
MRGPRX4 Q96LA9 1/20 0.58
GPR132 Q9UNW8 1/20 0.58
ALDH1A1 P00352 1/20 0.58
FAAH O00519 1/20 0.57
CNR2 P34972 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30412560 1.00 NR4A2 (0.77) NR4A2MAOBSMPD1SRD5A2PTPN1
SCHEMBL8193954 0.88 NR4A2 (0.72) NR4A2MAOBSMPD1SRD5A2PTPN1
SCHEMBL1795022 0.87 MEN1 (0.75) NR4A2MAOBSMPD1SRD5A2PTPN1
SCHEMBL26574732 0.87 MEN1 (0.70) NR4A2MAOBSMPD1SRD5A2PTPN1
SCHEMBL339009 0.87 NR4A2 (1.00) NR4A2MAOBSMPD1SRD5A2PTPN1
SCHEMBL30207018 0.87 NR4A2 (1.00) NR4A2MAOBSMPD1SRD5A2PTPN1
SCHEMBL7908051 0.87 SRD5A2 (0.85) NR4A2MAOBSMPD1SRD5A2PTPN1
SCHEMBL2928585 0.86 NR4A2 (0.58) NR4A2MAOBSMPD1SRD5A2PTPN1
Hydrochloric Acid SCHEMBL4748074 0.85 NR4A2 (0.97) NR4A2MAOBSMPD1SRD5A2PTPN1
SCHEMBL3442746 0.85 NR4A2 (0.79) NR4A2MAOBSMPD1SRD5A2PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 139 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3002280-B1 CYCLIC TRIAZO AND DIAZO SODIUM CHANNEL BLOCKERS UNIV GREENWICH (GB) 2023-05-24 EP disclosed
US-11345676-B2 Apoptosis signal-regulating kinase 1 (ASK 1) inhibitor compounds PHARMAKEA, INC. (US) 2022-05-31 US disclosed
US-11345676-B2 Apoptosis signal-regulating kinase 1 (ASK 1) inhibitor compounds PHARMAKEA, INC. (US) 2022-05-31 US disclosed
US-11072576-B2 Compositions and methods for glucose transport inhibition OHIO UNIVERSITY (US) 2021-07-27 US disclosed
US-20210017166-A1 PHARMACOKINETICALLY IMPROVED COMPOUNDS SURFACE LOGIX LLC (US) 2021-01-21 US disclosed
US-10570123-B2 Pharmacokinetically improved compounds SURFACE LOGIX, LLC (US) 2020-02-25 US disclosed
US-20200048218-A1 APOPTOSIS SIGNAL-REGULATING KINASE 1 (ASK 1) INHIBITOR COMPOUNDS PHARMAKEA, INC. 2020-02-13 US disclosed
US-20200048218-A1 APOPTOSIS SIGNAL-REGULATING KINASE 1 (ASK 1) INHIBITOR COMPOUNDS PHARMAKEA, INC. 2020-02-13 US disclosed
EP-3601250-A1 APOPTOSIS SIGNAL-REGULATING KINASE 1 (ASK 1) INHIBITOR COMPOUNDS Pharmakea, Inc. (US) 2020-02-05 EP disclosed
US-20190345094-A1 COMPOSITIONS AND METHODS FOR GLUCOSE TRANSPORT INHIBITION OHIO UNIVERSITY 2019-11-14 US disclosed
EP-0629232-A1 FUEL ADDITIVE COMPOSITIONS CONTAINING POLY(OXYALKYLENE) HYDROXYAROMATIC ESTERS AND ALIPHATIC AMINES CHEVRON CHEMICAL COMPANY (US) 1994-12-21 EP disclosed
EP-0626994-A1 FUEL ADDITIVE COMPOSITIONS CONTAINING POLY(OXYALKYLENE) HYDROXYAROMATIC ESTERS AND POLY(OXYALKYLENE) AMINES CHEVRON CHEMICAL COMPANY (US) 1994-12-07 EP disclosed
US-5366519-A Antideposit agents for fuels CHEVRON RESEARCH AND TECHNOLOGY COMPANY (US) 1994-11-22 US disclosed
WO-1994020062-A2 BALANOIDS AS PROTEIN KINASE C INHIBITORS ELI LILLY AND COMPANY (US) 1994-09-15 WO disclosed
WO-1994014926-A1 POLY(OXYALKYLENE) HYDROXYAROMATIC ESTERS AND FUEL COMPOSITIONS CONTAINING THE SAME CHEVRON RESEARCH AND TECHNOLOGY COMPANY (US) 1994-07-07 WO disclosed
WO-1994014928-A1 FUEL ADDITIVE COMPOSITIONS CONTAINING POLY(OXYALKYLENE) HYDROXYAROMATIC ESTERS AND ALIPHATIC AMINES CHEVRON RESEARCH AND TECHNOLOGY COMPANY (US) 1994-07-07 WO disclosed
WO-1994014930-A1 FUEL ADDITIVE COMPOSITIONS CONTAINING POLY(OXYALKYLENE) HYDROXYAROMATIC ESTERS AND POLY(OXYALKYLENE) AMINES CHEVRON RESEARCH AND TECHNOLOGY COMPANY (US) 1994-07-07 WO disclosed
US-5223510-A ALKYLAMINOALKYL DERIVATIVES OF BENZOFURAN, BENZOTHIOPHENE, INDOLE AND INDOLIZINE, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM SANOFI (FR) 1993-06-29 US disclosed
EP-0135838-A2 3-Phenyl-4-methoxycarbonyl pyrazoles, process for their preparation and their use against plant growth BASF Aktiengesellschaft (DE) 1985-04-03 EP disclosed
EP-0051828-B1 N-BENZOYL-ALPHA-ANILINO ALKANE CARBOXYLIC ACIDS, SALTS AND ESTERS THEREOF, PROCESS FOR PRODUCING THE SAME AND PHARMACEUTICAL PREPARATIONS CONTAINING THE SAME A. Nattermann & Cie. GmbH (DE) 1984-03-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190345094-A1 COMPOSITIONS AND METHODS FOR GLUCOSE TRANSPORT INHIBITION SLC2A1, SLC2A4, SLC2A3 NR4A2 803/4885MAOB 4311/4885SMPD1 1677/4885
US-11072576-B2 Compositions and methods for glucose transport inhibition SLC2A1, SLC2A4, SLC2A3 NR4A2 803/4885MAOB 4311/4885SMPD1 1677/4885
US-20210017166-A1 PHARMACOKINETICALLY IMPROVED COMPOUNDS ROCK2, ROCK1, RHOT2 NR4A2 4610/4885MAOB 1336/4885SMPD1 73/4885
US-20200048218-A1 APOPTOSIS SIGNAL-REGULATING KINASE 1 (ASK 1) INHIBITOR COMPOUNDS BAX, BAD, BCL2 NR4A2 2830/4885MAOB 4327/4885SMPD1 1892/4885
US-10570123-B2 Pharmacokinetically improved compounds ROCK2, ROCK1, RHOT2 NR4A2 4610/4885MAOB 1336/4885SMPD1 73/4885
US-11345676-B2 Apoptosis signal-regulating kinase 1 (ASK 1) inhibitor compounds BAX, BAD, BCL2 NR4A2 2830/4885MAOB 4327/4885SMPD1 1892/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.