SCHEMBL3401392

SCHEMBL3401392

CCCCc1cc(OC)c(C(=O)N2CCN(CC)CC2)s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.44
ALDH1A1 P00352 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
MEN1 O00255 3/20 0.43
HPGD P15428 2/20 0.43
KDM4E B2RXH2 2/20 0.43
GAA P10253 2/20 0.43
HTT P42858 1/20 0.43
MAPK1 P28482 1/20 0.43
HSD17B10 Q99714 1/20 0.43
NPC1 O15118 3/20 0.42
RAB9A P51151 2/20 0.42
MKNK2 Q9HBH9 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MAPT P10636 1/20 0.41
PTPN7 P35236 1/20 0.40
DUSP3 P51452 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
DRD2 P14416 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3400976 0.81 KMT2A (0.50) KMT2AALDH1A1SMN1; SMN2MEN1HPGD
SCHEMBL16233183 0.71 ALDH1A1 (0.54) KMT2AALDH1A1SMN1; SMN2MEN1HPGD
SCHEMBL10447618 0.69 ALDH1A1 (0.70) ALDH1A1SMN1; SMN2KDM4EGAAL3MBTL1
SCHEMBL3400265 0.66 HTR2C (0.46) KMT2AALDH1A1SMN1; SMN2MEN1HPGD
SCHEMBL7879085 0.66 ALDH1A1 (0.53) KMT2AALDH1A1SMN1; SMN2MEN1HPGD
SCHEMBL8322979 0.66 DRD2 (0.70) ALDH1A1HPGDKDM4EL3MBTL1DRD2
SCHEMBL15649918 0.65 ALDH1A1 (0.57) KMT2AALDH1A1SMN1; SMN2MEN1HPGD
SCHEMBL22172135 0.65 ALDH1A1 (0.52) KMT2AALDH1A1MEN1HPGDKDM4E
SCHEMBL4283460 0.64 ALDH1A1 (0.58) KMT2AALDH1A1SMN1; SMN2MEN1KDM4E
SCHEMBL10282569 0.64 MEN1 (0.70) KMT2AALDH1A1SMN1; SMN2MEN1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247588-A2 FUSED HETEROCYCLIC DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2010-11-10 EP disclosed
WO-2009107850-A2 FUSED HETEROCYCLIC DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-09-03 WO disclosed