SCHEMBL3400976

SCHEMBL3400976

CCN1CCN(C(=O)c2sc(C)cc2OC)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.50
ALDH1A1 P00352 6/20 0.47
MEN1 O00255 3/20 0.47
HPGD P15428 2/20 0.47
GAA P10253 2/20 0.47
KDM4E B2RXH2 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HTT P42858 1/20 0.47
MAPK1 P28482 1/20 0.47
HSD17B10 Q99714 1/20 0.47
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
TDP1 Q9NUW8 1/20 0.45
MKNK2 Q9HBH9 1/20 0.45
MAPT P10636 1/20 0.45
PTPN7 P35236 1/20 0.44
DUSP3 P51452 1/20 0.44
POLB P06746 1/20 0.43
CYP2C19 P33261 1/20 0.43
PARP1 P09874 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3401392 0.81 KMT2A (0.44) KMT2AALDH1A1MEN1HPGDGAA
SCHEMBL3401052 0.73 CYP2C9 (0.65) KMT2AMEN1SMN1; SMN2NPC1POLB
SCHEMBL10447618 0.73 ALDH1A1 (0.70) ALDH1A1GAAKDM4ESMN1; SMN2POLB
SCHEMBL3397115 0.73 SMN1; SMN2 (0.56) KMT2AALDH1A1MEN1HPGDKDM4E
SCHEMBL7879085 0.73 ALDH1A1 (0.53) KMT2AALDH1A1MEN1HPGDGAA
SCHEMBL3400265 0.73 HTR2C (0.46) KMT2AALDH1A1MEN1HPGDGAA
SCHEMBL3402191 0.71 TP53 (0.45) KMT2AALDH1A1MEN1HPGDGAA
SCHEMBL18823273 0.70 ALDH1A1 (0.58) KMT2AALDH1A1MEN1HPGDGAA
SCHEMBL8322979 0.70 DRD2 (0.70) ALDH1A1HPGDKDM4EL3MBTL1LMNA
SCHEMBL22172135 0.69 ALDH1A1 (0.52) KMT2AALDH1A1MEN1HPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247588-A2 FUSED HETEROCYCLIC DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2010-11-10 EP disclosed
WO-2009107850-A2 FUSED HETEROCYCLIC DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-09-03 WO disclosed