SCHEMBL3409749

SCHEMBL3409749

COc1cc(Nc2nc(C(F)(F)F)cc(C(F)(F)F)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 7/20 0.42
KCNH2 Q12809 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
ABCB1 P08183 1/20 0.40
ABCC1 P33527 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
ULK1 O75385 1/20 0.39
ULK2 Q8IYT8 1/20 0.39
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
PSEN1 P49768 1/20 0.37
PSEN2 P49810 1/20 0.37
APH1B Q8WW43 1/20 0.37
NCSTN Q92542 1/20 0.37
APH1A Q96BI3 1/20 0.37
PSENEN Q9NZ42 1/20 0.37
DOT1L Q8TEK3 1/20 0.37
AURKA O14965 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3405216 0.96 IMPDH2 (0.39) IMPDH2KCNH2NPC1RAB9AABCB1
SCHEMBL3406095 0.91 CYP3A4 (0.44) IMPDH2KCNH2NPC1RAB9AABCB1
SCHEMBL3406878 0.89 SYK (0.50) SYK
SCHEMBL3407100 0.87 MAPT (0.48) LMNAMAPTMAPK1PTGS2
SCHEMBL3410260 0.87 NPC1 (0.53) IMPDH2KCNH2NPC1RAB9AABCG2
SCHEMBL3406812 0.87 IMPDH2 (0.39) IMPDH2ULK1ULK2LMNAMAPT
SCHEMBL3406884 0.86 TLR8 (0.56) IMPDH2LMNAMAPTMAPK1
SCHEMBL3410560 0.85 NPC1 (0.37) IMPDH2KCNH2NPC1RAB9AABCG2
SCHEMBL3410316 0.85 IMPDH2 (0.44) IMPDH2KCNH2NPC1RAB9AABCG2
SCHEMBL3406378 0.84 PTGS2 (0.42) IMPDH2LMNAMAPTPTGS2SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed