SCHEMBL3404604

SCHEMBL3404604

CCN(NC(=O)Oc1ccc(OC(=O)c2csc(NC(C)=O)n2)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.42
SMN1; SMN2 Q16637 9/20 0.41
RAB9A P51151 7/20 0.41
MAPT P10636 2/20 0.41
HSP90AA1 P07900 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPC1 O15118 5/20 0.39
LMNA P02545 4/20 0.38
GLA P06280 1/20 0.38
ABCB1 P08183 1/20 0.38
ALDH1A1 P00352 2/20 0.37
CASP3 P42574 1/20 0.37
HTT P42858 1/20 0.37
SENP8 Q96LD8 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
PIM1 P11309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3406288 0.85 NPC1 (0.58) SMN1; SMN2RAB9AMAPTMAPK1NPC1
SCHEMBL3401758 0.84 AOC3 (0.54) SMN1; SMN2RAB9ANPC1LMNAALDH1A1
SCHEMBL3404608 0.83 SMN1; SMN2 (0.43) L3MBTL1SMN1; SMN2RAB9AMAPTHSP90AA1
SCHEMBL3404610 0.80 SMN1; SMN2 (0.48) L3MBTL1SMN1; SMN2RAB9AMAPTHSP90AA1
SCHEMBL3406052 0.77 AOC3 (0.49) SMN1; SMN2RAB9ANPC1LMNAALDH1A1
SCHEMBL973157 0.77 AOC3 (0.41) L3MBTL1SMN1; SMN2RAB9AMAPTHSP90AA1
SCHEMBL3407934 0.76 MEN1 (0.41) SMN1; SMN2MAPTGLAALDH1A1HTT
SCHEMBL3401395 0.75 MAPT (0.40) SMN1; SMN2RAB9AMAPTNPC1GLA
SCHEMBL972198 0.75 AOC3 (0.39) L3MBTL1SMN1; SMN2RAB9AMAPTHSP90AA1
SCHEMBL3404977 0.71 MGLL (0.51) SMN1; SMN2RAB9AMAPTCYP1A2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2252604-A1 THIAZOLE DERIVATIVE AND USE THEREOF AS VAP-1 INHIBITOR R-Tech Ueno, Ltd. (JP) 2010-11-24 EP disclosed
WO-2009096609-A1 THIAZOLE DERIVATIVE AND USE THEREOF AS VAP-1 INHIBITOR R-TECH UENO, LTD. (JP) 2009-08-06 WO disclosed