SCHEMBL3407934

SCHEMBL3407934

CCN(NC(=O)Oc1ccc(O)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
BCHE P06276 3/20 0.40
CHRM2 P08172 3/20 0.40
ELANE P08246 6/20 0.39
MIF P14174 1/20 0.38
AKT1 P31749 2/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
THRB P10828 1/20 0.38
BLM P54132 1/20 0.38
CASP6 P55212 1/20 0.38
GFER P55789 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
NQO2 P16083 1/20 0.37
HTT P42858 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3401395 0.88 MAPT (0.40) MEN1KMT2ABCHECHRM2ELANE
SCHEMBL3404977 0.84 MGLL (0.51) KMT2AMAPTGAASMN1; SMN2ALDH1A1
SCHEMBL3406288 0.77 NPC1 (0.58) MEN1KMT2AMAPTKDM4EGAA
SCHEMBL3404604 0.76 L3MBTL1 (0.42) MAPTKDM4EGLATDP1HTT
SCHEMBL3401758 0.74 AOC3 (0.54) HTTSMN1; SMN2ALDH1A1
SCHEMBL3407932 0.73 HTT (0.47) MEN1KMT2ABCHECHRM2ELANE
SCHEMBL10866251 0.70 MAPT (0.46) KMT2AELANEMIFMAPTKDM4E
SCHEMBL4057059 0.69 ELANE (0.70) MEN1KMT2AELANEMIFMAPT
SCHEMBL27774480 0.69 MEN1 (0.53) MEN1KMT2ABCHECHRM2ELANE
SCHEMBL3894800 0.69 TSHR (0.42) CHRM2MIFMAPTKDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2252604-A1 THIAZOLE DERIVATIVE AND USE THEREOF AS VAP-1 INHIBITOR R-Tech Ueno, Ltd. (JP) 2010-11-24 EP disclosed
WO-2009096609-A1 THIAZOLE DERIVATIVE AND USE THEREOF AS VAP-1 INHIBITOR R-TECH UENO, LTD. (JP) 2009-08-06 WO disclosed