SCHEMBL3406053

SCHEMBL3406053

CN(Cc1ccccc1)C(=O)OC1(c2ccccc2)CCC2(CC1)OCCO2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA4 P43681 1/20 0.40
HPGD P15428 4/20 0.39
TSHR P16473 3/20 0.39
ALDH1A1 P00352 2/20 0.39
GAA P10253 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
C5AR1 P21730 1/20 0.39
KMT2A Q03164 3/20 0.38
MEN1 O00255 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRL1 P41146 1/20 0.37
RIPK1 Q13546 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3413550 0.84 OPRM1 (0.40) HPGDTSHRALDH1A1GAAOPRM1
SCHEMBL3413530 0.80 ALDH1A1 (0.42) NPC1RAB9AHPGDTSHRALDH1A1
SCHEMBL4353815 0.79 HSD11B1 (0.48) NPC1RAB9ACA12CA9HPGD
SCHEMBL6938953 0.73 OPRM1 (0.45) RAB9ATSHRALDH1A1SMN1; SMN2KMT2A
SCHEMBL4152236 0.71 ALDH1A1 (0.34) NPC1RAB9ATSHRALDH1A1GAA
SCHEMBL6132327 0.70 OPRM1 (0.47) TSHRALDH1A1GAAOPRM1OPRL1
SCHEMBL3413377 0.69 SLC6A4 (0.47) TSHRALDH1A1SMN1; SMN2C5AR1OPRM1
SCHEMBL3232238 0.69 CYP2C19 (0.46) TSHRALDH1A1KMT2AMEN1
Oxalic Acid SCHEMBL7908190 0.68 C5AR1 (0.54) TSHRC5AR1OPRM1LMNA
SCHEMBL1668104 0.68 LMNA (0.56) NPC1RAB9AALDH1A1GAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2502907-B1 Substituted 4-aminocyclohexane derivatives GRUENENTHAL GMBH (DE) 2018-08-29 EP disclosed
EP-2518052-B1 Substituted 4-aminocyclohexane derivatives GRUENENTHAL GMBH (DE) 2017-12-20 EP disclosed
EP-2260021-B1 SUBSTITUTED 4-AMINOCYCLOHEXANE DERIVATIVES GRUENENTHAL GMBH (DE) 2014-04-23 EP disclosed
EP-2518052-A1 Substituted 4-aminocyclohexane derivatives Grünenthal GmbH (DE) 2012-10-31 EP disclosed
EP-2502907-A1 Substituted 4-aminocyclohexane derivatives Grünenthal GmbH (DE) 2012-09-26 EP disclosed
EP-2260021-A1 SUBSTITUTED 4-AMINOCYCLOHEXANE DERIVATIVES Grünenthal GmbH (DE) 2010-12-15 EP disclosed
WO-2009118168-A1 SUBSTITUTED 4-AMINOCYCLOHEXANE DERIVATIVES Grünenthal GmbH (DE) 2009-10-01 WO disclosed