SCHEMBL3406436

SCHEMBL3406436

COc1cc(Nc2nc(CC=O)cc(-c3ccc(C(F)(F)F)cc3)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 2/20 0.35
PTGS2 P35354 2/20 0.35
IMPDH2 P12268 3/20 0.35
ACP1 P24666 1/20 0.34
TDO2 P48775 1/20 0.34
PSEN1 P49768 2/20 0.34
PSEN2 P49810 2/20 0.34
APH1B Q8WW43 2/20 0.34
NCSTN Q92542 2/20 0.34
APH1A Q96BI3 2/20 0.34
PSENEN Q9NZ42 2/20 0.34
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
GAK O14976 1/20 0.33
DHODH Q02127 1/20 0.33
CDK9 P50750 2/20 0.33
CCNT1 O60563 1/20 0.33
KCNH2 Q12809 1/20 0.33
CDK2 P24941 1/20 0.33
JAK2 O60674 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3412354 0.83 PTGS2 (0.39) PLK1PTGS2IMPDH2ACP1TDO2
SCHEMBL3410261 0.83 SYK (0.37) TDO2ROCK2ROCK1DHODH
SCHEMBL3413279 0.82 CDK2 (0.46) CDK9CCNT1CDK2JAK2
SCHEMBL3408556 0.79 PLK1 (0.36) PLK1PTGS2IMPDH2ACP1TDO2
SCHEMBL3407100 0.79 MAPT (0.48) PTGS2CDK2JAK2
SCHEMBL3411225 0.77 MTTP (0.41) IMPDH2
SCHEMBL3410530 0.77 PLK1 (0.46) PLK1PSEN1PSEN2APH1BNCSTN
SCHEMBL3412730 0.77 PIK3CA (0.40) IMPDH2PSEN1PSEN2APH1BNCSTN
SCHEMBL3409749 0.77 IMPDH2 (0.42) PLK1PTGS2IMPDH2PSEN1PSEN2
SCHEMBL3410226 0.76 PLK1 (0.47) PLK1CDK9CCNT1CDK2JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed