SCHEMBL3406844

SCHEMBL3406844

COc1cc(Nc2nc(C)cc(N3CCCCC3)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GALR2 O43603 11/20 0.48
SLC2A1 P11166 3/20 0.48
GALR1 P47211 2/20 0.48
MEN1 O00255 2/20 0.45
ALDH1A1 P00352 2/20 0.45
KMT2A Q03164 2/20 0.45
KDM4E B2RXH2 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
ALOX15 P16050 1/20 0.45
NR4A1 P22736 1/20 0.45
MAPK1 P28482 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
AURKA O14965 1/20 0.44
AURKB Q96GD4 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTT P42858 1/20 0.43
EHMT2 Q96KQ7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3411061 0.99 SLC2A1 (0.48) GALR2SLC2A1GALR1MEN1ALDH1A1
SCHEMBL3413403 0.91 IMPDH2 (0.49) SLC2A1MEN1ALDH1A1KMT2AKDM4E
SCHEMBL3411892 0.91 SLC2A1 (0.43) GALR2SLC2A1GALR1MEN1ALDH1A1
SCHEMBL3412580 0.89 GALR2 (0.44) GALR2SLC2A1GALR1KDM4EMAPT
SCHEMBL3409900 0.88 AURKA (0.47) GALR2SLC2A1GALR1AURKAAURKB
SCHEMBL3410528 0.88 GALR2 (0.42) GALR2SLC2A1GALR1MEN1ALDH1A1
SCHEMBL3410260 0.86 NPC1 (0.53) MEN1ALDH1A1KMT2AKDM4EGAA
SCHEMBL3410125 0.82 GALR2 (0.51) GALR2GALR1KDM4EMAPTMAPK1
SCHEMBL3406068 0.82 NPC1 (0.46) MEN1ALDH1A1KMT2AKDM4EMAPT
SCHEMBL3407955 0.81 NPC1 (0.51) MEN1KMT2AKDM4EGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed