SCHEMBL3409900

SCHEMBL3409900

COc1cc(Nc2nc(C)cc(N3CCN(S(C)(=O)=O)CC3)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AURKA O14965 8/20 0.47
AURKB Q96GD4 2/20 0.45
SLC2A1 P11166 3/20 0.42
BRD4 O60885 1/20 0.39
SUV39H2 Q9H5I1 1/20 0.38
PDE7A Q13946 1/20 0.38
GALR2 O43603 2/20 0.38
GALR1 P47211 1/20 0.38
JAK2 O60674 1/20 0.37
JAK3 P52333 1/20 0.37
ALK Q9UM73 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3411061 0.89 SLC2A1 (0.48) AURKAAURKBSLC2A1BRD4GALR2
SCHEMBL3406844 0.88 GALR2 (0.48) AURKAAURKBSLC2A1BRD4GALR2
SCHEMBL3413403 0.85 IMPDH2 (0.49) AURKAAURKBSLC2A1BRD4JAK2
SCHEMBL3411892 0.85 SLC2A1 (0.43) AURKAAURKBSLC2A1BRD4PDE7A
SCHEMBL3410260 0.81 NPC1 (0.53) BRD4
SCHEMBL4090603 0.79 PSEN1 (0.51) AURKA
SCHEMBL3410528 0.79 GALR2 (0.42) AURKAAURKBSLC2A1GALR2GALR1
SCHEMBL3412580 0.78 GALR2 (0.44) AURKAAURKBSLC2A1GALR2GALR1
SCHEMBL3406068 0.77 NPC1 (0.46) BRD4
SCHEMBL3407955 0.76 NPC1 (0.51) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed