SCHEMBL3407932

SCHEMBL3407932

CCOC(=O)N(NC(=O)Oc1ccc(O)cc1)C(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.47
BCHE P06276 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CHRM2 P08172 1/20 0.40
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CA9 Q16790 2/20 0.40
CA14 Q9ULX7 2/20 0.40
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
ELANE P08246 4/20 0.39
MIF P14174 1/20 0.38
PRTN3 P24158 1/20 0.38
KDM4E B2RXH2 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
THRB P10828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3401402 0.88 HTT (0.46) HTTSMN1; SMN2KDM4EGLAGAA
SCHEMBL3404972 0.84 MGLL (0.51) HTTBCHESMN1; SMN2CA1CA2
SCHEMBL3404315 0.76 CA12 (0.52) SMN1; SMN2CA12CA1CA2CA7
SCHEMBL3401766 0.74 AOC3 (0.54) HTTSMN1; SMN2MAPTLMNAALDH1A1
SCHEMBL3407934 0.73 MEN1 (0.41) HTTBCHESMN1; SMN2CHRM2ELANE
SCHEMBL8536318 0.69 CA2 (0.55) SMN1; SMN2CA12CA1CA2CA7
SCHEMBL27774480 0.69 MEN1 (0.53) HTTBCHESMN1; SMN2CHRM2ELANE
SCHEMBL9714370 0.69 CYP3A4 (0.55) HTTSMN1; SMN2KDM4EGAAMAPT
SCHEMBL9651163 0.68 MGAM (0.34) SMN1; SMN2GAAMAPTKMT2AMEN1
SCHEMBL25407106 0.68 ELANE (0.51) BCHECA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2252604-A1 THIAZOLE DERIVATIVE AND USE THEREOF AS VAP-1 INHIBITOR R-Tech Ueno, Ltd. (JP) 2010-11-24 EP disclosed
WO-2009096609-A1 THIAZOLE DERIVATIVE AND USE THEREOF AS VAP-1 INHIBITOR R-TECH UENO, LTD. (JP) 2009-08-06 WO disclosed