SCHEMBL3401402

SCHEMBL3401402

CCOC(=O)N(NC(=O)Oc1ccc(N)cc1)C(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.46
LMNA P02545 3/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
MAOA P21397 1/20 0.41
MAPT P10636 3/20 0.40
TDP1 Q9NUW8 2/20 0.40
KDM4E B2RXH2 1/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
THRB P10828 1/20 0.40
BLM P54132 1/20 0.40
CASP6 P55212 1/20 0.40
GFER P55789 1/20 0.40
PPIB P23284 1/20 0.39
PPIA P62937 1/20 0.39
PPID Q08752 1/20 0.39
PPIG Q13427 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.37
ABCB1 P08183 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3407932 0.88 HTT (0.47) HTTLMNAMAPTTDP1KDM4E
SCHEMBL3404972 0.83 MGLL (0.51) HTTCYP3A4MAPTGAASMN1; SMN2
SCHEMBL3401395 0.74 MAPT (0.40) HTTMAPTTDP1KDM4EGLA
SCHEMBL9195477 0.70 LMNA (0.56) HTTLMNACYP1A2CYP3A4MAOA
SCHEMBL29023046 0.70 LMNA (0.49) HTTLMNACYP1A2CYP3A4MAOA
SCHEMBL2493638 0.70 MEN1 (0.51) HTTLMNACYP1A2CYP3A4MAOA
SCHEMBL3813706 0.69 MAPT (0.51) HTTLMNAMAPTTDP1KDM4E
SCHEMBL13724309 0.69 KMT2A (0.52) MAPTTDP1KDM4EGLAGAA
Hydrochloric Acid SCHEMBL27454826 0.68 LMNA (0.50) HTTLMNACYP1A2CYP3A4MAOA
SCHEMBL9714370 0.68 CYP3A4 (0.55) HTTLMNACYP1A2CYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2252604-A1 THIAZOLE DERIVATIVE AND USE THEREOF AS VAP-1 INHIBITOR R-Tech Ueno, Ltd. (JP) 2010-11-24 EP disclosed
WO-2009096609-A1 THIAZOLE DERIVATIVE AND USE THEREOF AS VAP-1 INHIBITOR R-TECH UENO, LTD. (JP) 2009-08-06 WO disclosed