SCHEMBL3407960

SCHEMBL3407960

COc1cc(Nc2nc(C)cc(OCCC(F)(F)C(F)(F)F)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
EHMT2 Q96KQ7 6/20 0.35
EHMT1 Q9H9B1 6/20 0.35
IMPDH2 P12268 6/20 0.35
DOT1L Q8TEK3 1/20 0.34
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
ULK1 O75385 1/20 0.33
ULK2 Q8IYT8 1/20 0.33
USP2 O75604 1/20 0.32
ABCB1 P08183 1/20 0.32
ABCC1 P33527 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
TERT O14746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3406681 0.87 NPC1 (0.41) KCNH2NPC1RAB9AEHMT2EHMT1
SCHEMBL3410702 0.85 USP2 (0.45) KCNH2NPC1RAB9AEHMT2EHMT1
SCHEMBL3413227 0.84 HTR6 (0.46) KCNH2NPC1RAB9AEHMT2EHMT1
SCHEMBL3406068 0.84 NPC1 (0.46) KCNH2NPC1RAB9AEHMT2EHMT1
SCHEMBL3410260 0.81 NPC1 (0.53) KCNH2NPC1RAB9AEHMT2EHMT1
SCHEMBL3410316 0.79 IMPDH2 (0.44) KCNH2NPC1RAB9AEHMT2EHMT1
SCHEMBL3412265 0.79 ABCB1 (0.39) KCNH2NPC1RAB9AIMPDH2DOT1L
SCHEMBL3413260 0.79 GAK (0.39) KCNH2NPC1RAB9AIMPDH2DOT1L
SCHEMBL3413137 0.79 CHRNA7 (0.40) KCNH2NPC1RAB9AEHMT2EHMT1
SCHEMBL3411085 0.79 NPC1 (0.42) KCNH2NPC1RAB9AEHMT2EHMT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed