SCHEMBL3410316

SCHEMBL3410316

COc1cc(OC)nc(Nc2ccc(-c3nc(C)c[nH]3)c(OC)c2)n1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 10/20 0.44
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
KCNH2 Q12809 1/20 0.40
DOT1L Q8TEK3 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.38
MAPT P10636 2/20 0.38
GAA P10253 1/20 0.38
TERT O14746 1/20 0.37
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
EHMT2 Q96KQ7 1/20 0.36
EHMT1 Q9H9B1 1/20 0.36
TP53 P04637 1/20 0.36
POLB P06746 1/20 0.36
RAD52 P43351 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3406068 0.95 NPC1 (0.46) IMPDH2NPC1RAB9AKCNH2DOT1L
SCHEMBL3410260 0.90 NPC1 (0.53) IMPDH2NPC1RAB9AKCNH2DOT1L
SCHEMBL3411085 0.86 NPC1 (0.42) IMPDH2NPC1RAB9AKCNH2DOT1L
SCHEMBL3410702 0.86 USP2 (0.45) IMPDH2NPC1RAB9AKCNH2DOT1L
SCHEMBL3409749 0.85 IMPDH2 (0.42) IMPDH2NPC1RAB9AKCNH2DOT1L
SCHEMBL3406662 0.85 NPC1 (0.40) IMPDH2NPC1RAB9AKCNH2DOT1L
SCHEMBL3408338 0.85 NPC1 (0.40) IMPDH2NPC1RAB9AKCNH2DOT1L
SCHEMBL3407955 0.85 NPC1 (0.51) IMPDH2NPC1RAB9AKCNH2DOT1L
SCHEMBL3406681 0.84 NPC1 (0.41) IMPDH2NPC1RAB9AKCNH2DOT1L
SCHEMBL3406468 0.82 KCNH2 (0.42) IMPDH2NPC1RAB9AKCNH2DOT1L

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed