SCHEMBL3408739

SCHEMBL3408739

Cc1c[nH]c(-c2ccc(Nc3nc(-c4ccc(C(F)(F)F)cc4)cc(C(C)(C)O)n3)cc2C)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.41
SYK P43405 3/20 0.38
CDK2 P24941 2/20 0.33
SLC1A3 P43003 1/20 0.33
SLC1A2 P43004 1/20 0.33
SLC1A1 P43005 1/20 0.33
MCHR1 Q99705 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
IDH2 P48735 1/20 0.33
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
IKBKB O14920 1/20 0.33
CHUK O15111 1/20 0.33
KDR P35968 1/20 0.32
TEK Q02763 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3406069 0.92 PTGS2 (0.40) PTGS2SYKCDK2MCHR1TP53
SCHEMBL3412354 0.90 PTGS2 (0.39) PTGS2SYKTP53MAPTPSEN1
SCHEMBL3409722 0.79 PIK3CA (0.41) PTGS2CDK2TP53MAPTPSEN1
SCHEMBL3408075 0.78 PSEN1 (0.47) PTGS2SYKMCHR1PSEN1PSEN2
SCHEMBL3405215 0.77 KCNH2 (0.37) PTGS2CDK2
SCHEMBL3409955 0.75 CDK2 (0.48) SYKCDK2IKBKBCHUKGSK3B
SCHEMBL3407100 0.74 MAPT (0.48) PTGS2CDK2TP53MAPT
SCHEMBL3413279 0.74 CDK2 (0.46) CDK2IKBKBCHUKGSK3B
SCHEMBL3408556 0.74 PLK1 (0.36) PTGS2SYKMAPTPSEN1PSEN2
SCHEMBL3410261 0.74 SYK (0.37) SYKTP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP claimed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO claimed
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed